SCHEMBL10114640

SCHEMBL10114640

CS(=O)(=O)Nc1cnc(NC(=O)c2ccc(C(F)(F)F)cc2O)s1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 2/20 0.43
USP2 O75604 6/20 0.41
USP8 P40818 6/20 0.41
TRPV1 Q8NER1 2/20 0.41
SCD O00767 1/20 0.39
SORT1 Q99523 2/20 0.39
P2RX1 P51575 2/20 0.39
P2RX4 Q99571 1/20 0.39
P2RX7 Q99572 1/20 0.39
TMPRSS4 Q9NRS4 1/20 0.39
NCS1 P62166 1/20 0.38
CSF1R P07333 1/20 0.38
POLQ O75417 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4757381 0.84 STAT3 (0.60) STAT3POLQMEN1KMT2A
SCHEMBL10114076 0.81 S1PR1 (0.44) STAT3USP2USP8TRPV1SCD
SCHEMBL4757379 0.81 STAT3 (0.56) STAT3MEN1KMT2A
SCHEMBL4757387 0.77 KCNMA1 (0.54) STAT3P2RX1P2RX4P2RX7TMPRSS4
SCHEMBL4757380 0.75 STAT3 (0.46) STAT3POLQMEN1KMT2A
SCHEMBL10114726 0.74 NPC1 (0.37) STAT3TRPV1CSF1RPOLQMEN1
SCHEMBL4757467 0.69 NPC1 (0.39) STAT3CSF1RPOLQMEN1KMT2A
SCHEMBL4757479 0.69 KCNMA1 (0.46) STAT3POLQMEN1KMT2A
SCHEMBL4755924 0.68 STAT3 (0.63) STAT3MEN1KMT2A
SCHEMBL5836220 0.68 CDK2 (0.56) STAT3SCDSORT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895752-B2 Alkylsulfonyl-substituted thiazolide compounds ROMARK LABORATORIES L.C. (US) 2014-11-25 US disclosed
US-8124632-B2 Alkylsulfonyl-substituted thiazolide compounds ROMARK LABORATORIES, L.C. (US) 2012-02-28 US disclosed
US-20090036467-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS ROMARK LABORATORIES L.C. 2009-02-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090036467-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS HAVCR2, EIF2AK2, AADAC STAT3 63/4885USP2 3480/4885USP8 2111/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.