SCHEMBL10117873

SCHEMBL10117873

Cc1ccc(-c2cnc(N)n2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 11/20 0.41
NR1H3 Q13133 3/20 0.38
MAPT P10636 2/20 0.38
GPR119 Q8TDV5 1/20 0.37
IKBKB O14920 1/20 0.37
USP2 O75604 1/20 0.36
TP53 P04637 1/20 0.36
MAPK1 P28482 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
MMP13 P45452 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
IDO1 P14902 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4062460 0.88 GABRG2 (0.45) NR1H2NR1H3MAPTGPR119USP2
SCHEMBL10117534 0.88 NR1H2 (0.40) NR1H2NR1H3MAPTUSP2TP53
SCHEMBL13663125 0.88 CYP1A2 (0.49) NR1H2NR1H3
SCHEMBL13655089 0.82 NR1H2 (0.38) NR1H2NR1H3MAPTGABRG2GABRB3
SCHEMBL4066085 0.81 FYN (0.43) NR1H2NR1H3GABRG2GABRB3GABRA5
SCHEMBL4239418 0.79 GABRG2 (0.44) NR1H2NR1H3GABRG2GABRB3GABRA5
SCHEMBL4058194 0.78 PTPN1 (0.55) MEN1KMT2A
SCHEMBL4242491 0.78 GABRG2 (0.38) NR1H2NR1H3GABRG2GABRB3GABRA5
SCHEMBL4237117 0.77 SMARCA2 (0.40) NR1H2NR1H3GPR119GABRG2GABRB3
SCHEMBL15707574 0.76 SCN3A (0.42) MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087976-A2 NOVEL INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2012-06-28 WO disclosed