SCHEMBL10117534

SCHEMBL10117534

CC(C)(C)OC(=O)n1c(-c2ccc(Br)cc2)cnc1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 10/20 0.40
NR1H3 Q13133 3/20 0.38
MAPT P10636 2/20 0.37
IDO1 P14902 1/20 0.36
DHFR P00374 1/20 0.36
EGFR P00533 1/20 0.36
ERBB2 P04626 1/20 0.36
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
MAPK1 P28482 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NTRK1 P04629 1/20 0.35
PIM1 P11309 1/20 0.35
ACVR1 Q04771 1/20 0.35
ABL1 P00519 1/20 0.35
BCR P11274 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10117873 0.88 NR1H2 (0.41) NR1H2NR1H3MAPTIDO1USP2
SCHEMBL4062460 0.87 GABRG2 (0.45) NR1H2NR1H3MAPTUSP2TP53
SCHEMBL13663125 0.86 CYP1A2 (0.49) NR1H2NR1H3NTRK1PIM1ABL1
SCHEMBL13655089 0.81 NR1H2 (0.38) NR1H2NR1H3MAPTGABRG2GABRB3
SCHEMBL4066085 0.80 FYN (0.43) NR1H2NR1H3GABRG2GABRB3GABRA5
SCHEMBL10117875 0.78 NPC1 (0.35) NR1H2NR1H3IDO1DHFREGFR
SCHEMBL4239418 0.78 GABRG2 (0.44) NR1H2NR1H3GABRG2GABRB3GABRA5
SCHEMBL10117510 0.77 MEN1 (0.45) NR1H2IDO1DHFREGFRERBB2
SCHEMBL4058194 0.77 PTPN1 (0.55) MEN1KMT2AABL1
SCHEMBL4242491 0.77 GABRG2 (0.38) NR1H2NR1H3IDO1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087976-A2 NOVEL INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2012-06-28 WO disclosed