SCHEMBL10120229

SCHEMBL10120229

COC(=O)C1CNCCN1c1ccccc1[N+](=O)[O-]

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 2/20 0.48
ICAM1 P05362 2/20 0.48
ITGAL P20701 2/20 0.48
MAPT P10636 6/20 0.40
MMP1 P03956 1/20 0.39
MMP3 P08254 1/20 0.39
MMP7 P09237 1/20 0.39
MMP9 P14780 1/20 0.39
MMP13 P45452 1/20 0.39
KMT2A Q03164 3/20 0.38
HTT P42858 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 4/20 0.38
LMNA P02545 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ABCC4 O15439 1/20 0.38
PLIN1 O60240 1/20 0.38
CACNA1F O60840 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18600524 0.87 KMT2A (0.40) ITGB2ICAM1ITGALMAPTKMT2A
SCHEMBL30237864 0.82 ALDH1A1 (0.39) ITGB2ICAM1ITGALMAPTMMP1
SCHEMBL31013530 0.82 ALDH1A1 (0.39) ITGB2ICAM1ITGALMAPTMMP1
SCHEMBL8084718 0.82 SMN1; SMN2 (0.46) MAPTKMT2AMEN1ALDH1A1LMNA
SCHEMBL8404563 0.79 MAPT (0.42) MAPTKMT2AHTTMEN1ALDH1A1
SCHEMBL8587625 0.79 HTT (0.44) MAPTKMT2AHTTALDH1A1SMN1; SMN2
SCHEMBL21360310 0.77 SLC6A4 (0.47) MMP1MMP3MMP7MMP9MMP13
SCHEMBL16731889 0.77 SLC6A4 (0.47) MMP1MMP3MMP7MMP9MMP13
SCHEMBL15210112 0.77 KMT2A (0.44) KMT2AHTTMEN1ALDH1A1LMNA
SCHEMBL10120707 0.76 MAPT (0.41) ITGB2ICAM1ITGALMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8969573-B2 Compounds for the inhibition of cellular proliferation PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2015-03-03 US disclosed
US-8969573-B2 Compounds for the inhibition of cellular proliferation PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2015-03-03 US disclosed
US-20130178505-A1 Compounds for the Inhibition of Cellular Proliferation PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2013-07-11 US disclosed
US-20130178505-A1 Compounds for the Inhibition of Cellular Proliferation PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2013-07-11 US disclosed
WO-2012006068-A2 COMPOUNDS FOR THE INHIBITION OF CELLULAR PROLIFERATION PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130178505-A1 Compounds for the Inhibition of Cellular Proliferation MKI67, EIF2AK2, CDK2 ITGB2 3995/4885ICAM1 3781/4885ITGAL 4540/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.