SCHEMBL10121183

SCHEMBL10121183

C=C(NCc1ccc(Oc2ccc(F)cc2Cl)c(F)c1)C1(NC(=O)c2cncnc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 3/20 0.41
CXCR4 P61073 1/20 0.41
CNR1 P21554 2/20 0.39
MET P08581 2/20 0.38
CARM1 Q86X55 2/20 0.37
PRMT6 Q96LA8 2/20 0.37
SCN3A Q9NY46 1/20 0.36
PYGL P06737 1/20 0.35
METAP2 P50579 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL765808 0.92 BDKRB1 (0.48) BDKRB1CXCR4CNR1METCARM1
SCHEMBL764462 0.87 BDKRB1 (0.40) BDKRB1CXCR4CNR1
SCHEMBL10121140 0.87 BDKRB1 (0.41) BDKRB1CXCR4CNR1METL3MBTL1
SCHEMBL764468 0.85 BDKRB1 (0.48) BDKRB1CXCR4CNR1METCARM1
SCHEMBL12239074 0.84 BDKRB1 (0.49) BDKRB1CNR1METCARM1PRMT6
SCHEMBL765831 0.82 BDKRB1 (0.51) BDKRB1CXCR4CNR1METPYGL
SCHEMBL765522 0.82 BDKRB1 (0.50) BDKRB1CXCR4CNR1METCARM1
Hydrochloric Acid SCHEMBL2546804 0.81 BDKRB1 (0.49) BDKRB1CXCR4CNR1METCARM1
SCHEMBL10121221 0.79 BDKRB1 (0.47) BDKRB1CXCR4CNR1MET
SCHEMBL10121264 0.79 BDKRB1 (0.49) BDKRB1CXCR4CNR1METAP2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188254-B1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-03-21 EP disclosed