SCHEMBL764462

SCHEMBL764462

C=C(NCc1ccc(Oc2ccc(Cl)c(Cl)c2)c(F)c1)C1(NC(=O)c2cncnc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 3/20 0.40
CNR1 P21554 2/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.36
LMNA P02545 1/20 0.36
SCN9A Q15858 1/20 0.36
PLA2G7 Q13093 1/20 0.35
LIPG Q9Y5X9 1/20 0.35
IGFBP3 P17936 1/20 0.35
HTR2A P28223 2/20 0.35
SLC6A4 P31645 2/20 0.35
KCNH2 Q12809 2/20 0.35
CXCR4 P61073 1/20 0.35
SCD O00767 1/20 0.34
PTGER4 P35408 1/20 0.34
WDR5 P61964 1/20 0.34
ABL1 P00519 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10121221 0.92 BDKRB1 (0.47) BDKRB1CNR1PTGDR2LMNASCN9A
SCHEMBL10121140 0.92 BDKRB1 (0.41) BDKRB1CNR1CXCR4PTGER4
SCHEMBL10121183 0.87 BDKRB1 (0.41) BDKRB1CNR1CXCR4
SCHEMBL12239073 0.85 BDKRB1 (0.47) BDKRB1CNR1WDR5
SCHEMBL10121264 0.84 BDKRB1 (0.49) BDKRB1CNR1CXCR4PTGER4
SCHEMBL764420 0.81 BDKRB1 (0.48) BDKRB1CNR1CXCR4PTGER4
SCHEMBL765524 0.80 BDKRB1 (0.51) BDKRB1CNR1SCN9ACXCR4PTGER4
SCHEMBL12239072 0.80 BDKRB1 (0.51) BDKRB1CNR1CXCR4
SCHEMBL2547691 0.80 BDKRB1 (0.53) BDKRB1CNR1
SCHEMBL764501 0.80 BDKRB1 (0.49) BDKRB1CNR1PTGDR2LMNALIPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188254-B1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-03-21 EP disclosed