SCHEMBL10128526

SCHEMBL10128526

O=C1Nc2cc([N+](=O)[O-])ccc2CC12CC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 2/20 0.47
TDP2 O95551 1/20 0.46
CYP3A4 P08684 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
PGR P06401 3/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
AKR1B1 P15121 2/20 0.42
CAPN9 O14815 1/20 0.42
CASP3 P42574 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
ADRA2A P08913 1/20 0.41
PNMT P11086 1/20 0.41
OTUD7B Q6GQQ9 2/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26087941 0.88 CRBN (0.47) CRBNTDP2CYP3A4ALDH1A1CYP2C9
SCHEMBL260824 0.76 CRBN (0.53) CRBNTDP2CYP3A4CA12CA1
SCHEMBL2993057 0.74 TDP2 (0.67) TDP2CYP3A4ALDH1A1PGRCAPN9
SCHEMBL17252079 0.74 CMA1 (0.54) TDP2OTUD7B
SCHEMBL260822 0.74 TDP2 (0.47) CRBNTDP2CYP3A4CA12CA1
SCHEMBL495833 0.73 CA9 (0.56) CRBNTDP2CYP3A4PGRCA9
SCHEMBL30270534 0.73 CA9 (0.56) CRBNTDP2CYP3A4PGRCA9
SCHEMBL15578816 0.73 PGR (0.62) TDP2CYP3A4ALDH1A1CYP2C9CYP2C19
SCHEMBL3604126 0.72 TDP2 (0.48) TDP2CYP3A4AKR1B1CAPN9CASP3
SCHEMBL31491273 0.72 TDP2 (0.48) TDP2CYP3A4AKR1B1CAPN9CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814878-B1 SPIRO-2, 4-PYRIMIDINEDIAMINE COMPOUNDS AND THEIR USES RIGEL PHARMACEUTICALS INC (US) 2012-01-04 EP disclosed