SCHEMBL10130615

SCHEMBL10130615

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nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 8/20 0.65
PRKCE Q02156 2/20 0.51
PRKCQ Q04759 2/20 0.51
PRKCD Q05655 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3189263 0.88 PRKCA (0.51) PRKCAPRKCEPRKCQPRKCD
SCHEMBL10026292 0.88 PRKCA (0.50) PRKCAPRKCEPRKCQPRKCD
SCHEMBL6370166 0.88 PRKCA (0.50) PRKCAPRKCEPRKCQPRKCD
SCHEMBL5026886 0.87 PRKCA (0.60) PRKCAPRKCEPRKCQPRKCD
SCHEMBL10135101 0.83 PRKCA (0.47) PRKCAPRKCEPRKCQPRKCD
SCHEMBL822220 0.82 PRKCA (0.63) PRKCAPRKCEPRKCQPRKCD
SCHEMBL19300984 0.81 PRKCA (0.44) PRKCAPRKCEPRKCQPRKCD
SCHEMBL8384532 0.80 PRKCA (0.97) PRKCAPRKCEPRKCQPRKCD
Acetic Acid SCHEMBL8675242 0.80 PRKCA (0.56) PRKCAPRKCEPRKCQPRKCD
SCHEMBL19300629 0.80 PRKCA (0.56) PRKCAPRKCEPRKCQPRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2287305-B2 RNA interference mediated inhibition of gene expression using short interfering nucleic acid (siNA) SIRNA THERAPEUTICS INC (US) 2017-11-29 EP disclosed
US-20160053269-A1 RNA INTERFERENCE MEDIATED INHIBITION OF GENE EXPRESSION USING CHEMICALLY MODIFIED SHORT INTERFERING NUCLEIC ACID (siNA) BANK OF AMERICA, N.A. 2016-02-25 US disclosed
EP-1423406-B2 RNA INTERFERENCE MEDIATED INHIBITION OF GENE EXPRESSION USING SHORT INTERFERING NUCLEIC ACID (SINA) SIRNA THERAPEUTICS INC (US) 2015-11-25 EP disclosed
EP-2902406-A1 RNA interference mediated inhibition of gene expression using short interfering nucleic acid (siNA) Sirna Therapeutics, Inc. (US) 2015-08-05 EP disclosed
EP-2287305-B1 RNA interference mediated inhibition of gene expression using short interfering nucleic acid (siNA) SIRNA THERAPEUTICS INC (US) 2015-01-07 EP disclosed
US-20140288148-A1 RNA INTERFERENCE MEDIATED INHIBITION OF GENE EXPRESSION USING CHEMICALLY MODIFIED SHORT INTERFERING NUCLEIC ACID (siNA) SIRNA THERAPEUTICS INC (US) 2014-09-25 US disclosed
US-20130018082-A1 RNA INTERFERENCE MEDIATED INHIBITION OF GENE EXPRESSION USING CHEMICALLY MODIFIED SHORT INTERFERING NUCLEIC ACID (siNA) BANK OF AMERICA, N.A. 2013-01-17 US disclosed
US-8153778-B2 RNA interference mediated inhibition of vascular cell adhesion molecule (VCAM) gene expression using short interfering nucleic acid (siNA) MERCK SHARP & DOHME CORP. (US) 2012-04-10 US disclosed
US-8076472-B2 RNA interference mediated inhibition of muscarinic colinergic receptor gene expression using short interfering nucleic acid (siNA) MERCK SHARP & DOHME CORP. (US) 2011-12-13 US disclosed
US-8013146-B2 RNA interference mediated inhibition of matrix metalloproteinase 13 (MMP13) gene expression using short interfering nucleic acid (siNA) MERCK SHARP & DOHME CORP. (US) 2011-09-06 US disclosed
US-8008472-B2 RNA interference mediated inhibition of human immunodeficiency virus (HIV) gene expression using short interfering nucleic acid (siNA) MERCK SHARP & DOHME CORP. (US) 2011-08-30 US disclosed
US-8008473-B2 RNA interference mediated inhibition of TNF and TNF receptor gene expression using short interfering nucleic acid (siNA) BANK OF AMERICA, N.A. 2011-08-30 US disclosed
US-7985853-B2 RNA interference mediated inhibition of platelet derived growth factor (PDGF) and platelet derived growth factor receptor (PDGFR) gene expression using short interfering nucleic acid (siNA) MERCK SHARP & DOHME CORP. (US) 2011-07-26 US disclosed
US-7928219-B2 chemically modified nucleic acid molecule; cancer; carcinoma, neovascularization, diabetic retinopathy, neovascular glaucoma, myopic degeneration and other proliferative diseases, restenosis and polycystic kidney disease MERCK SHARP & DOHME CORP. (US) 2011-04-19 US disclosed
US-7928220-B2 for treating ocular disease, cancer and proliferative diseases and any other disease, condition, trait or indication that can respond to the level of SDF-1 in a cell or tissue MERCK SHARP & DOHME CORP. (US) 2011-04-19 US disclosed
US-7855284-B2 RNA interference mediated inhibition of checkpoint kinase-1 (CHK-1) gene expression using short interfering nucleic acid (siNA) SIRNA THERAPEUTICS, INC. (US) 2010-12-21 US disclosed
US-20090299045-A1 Cancer, inflammatory, respiratory, autoimmune, cardiovascular, neurological, and/or proliferative diseases SIRNA THERAPEUTICS, INC. (US) 2009-12-03 US disclosed
US-20090099119-A1 RNA INTERFERENCE MEDIATED INHIBITION OF RAS GENE EXPRESSION USING SHORT INTERFERING NUCLEIC ACID (siNA) SIRNA THERAPEUTICS, INC. (US) 2009-04-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090299045-A1 Cancer, inflammatory, respiratory, autoimmune, cardiovascular, neurological, and/or proliferative diseases IL15RA, IL23R, IL2RA PRKCA 3148/4885PRKCE 3900/4885PRKCQ 3942/4885
US-20130018082-A1 RNA INTERFERENCE MEDIATED INHIBITION OF GENE EXPRESSION USING CHEMICALLY MODIFIED SHORT INTERFERING NUCLEIC ACID (siNA) AGO2, SNRPE, SRRT PRKCA 2538/4885PRKCE 4524/4885PRKCQ 4317/4885
US-20090099119-A1 RNA INTERFERENCE MEDIATED INHIBITION OF RAS GENE EXPRESSION USING SHORT INTERFERING NUCLEIC ACID (siNA) KRAS, HRAS, NRAS PRKCA 884/4885PRKCE 1730/4885PRKCQ 1454/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.