SCHEMBL10135256

SCHEMBL10135256

c1ccc(Nc2nc3ccccc3c3ccccc23)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 3/20 0.67
CSNK2A1 P68400 1/20 0.64
ABCG2 Q9UNQ0 3/20 0.62
MEN1 O00255 2/20 0.62
KMT2A Q03164 2/20 0.62
PDE5A O76074 6/20 0.61
KDM1A O60341 1/20 0.59
CLK4 Q9HAZ1 3/20 0.56
MAPK14 Q16539 2/20 0.56
DAPK3 O43293 1/20 0.56
MAP4K4 O95819 1/20 0.56
ABL1 P00519 1/20 0.56
EGFR P00533 1/20 0.56
ERBB2 P04626 1/20 0.56
PIM1 P11309 1/20 0.56
PRKACA P17612 1/20 0.56
LTK P29376 1/20 0.56
MAPK8 P45983 1/20 0.56
CSNK1A1 P48729 1/20 0.56
RPS6KA3 P51812 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10131633 0.84 CSNK2A1 (0.67) NPY5RCSNK2A1ABCG2MEN1KMT2A
SCHEMBL13702755 0.84 CSNK2A1 (0.65) NPY5RCSNK2A1ABCG2MEN1KMT2A
SCHEMBL17740777 0.84 ABCG2 (0.57) CSNK2A1ABCG2MEN1KMT2APDE5A
SCHEMBL19261422 0.83 PDE5A (0.70) NPY5RCSNK2A1ABCG2MEN1KMT2A
SCHEMBL13903883 0.82 MEN1 (0.69) NPY5RABCG2MEN1KMT2APDE5A
SCHEMBL1755564 0.82 ALDH1A1 (0.48) NPY5RCSNK2A1ABCG2MEN1KMT2A
Hydrochloric Acid SCHEMBL1705655 0.80 ALDH1A1 (0.46) NPY5RCSNK2A1ABCG2MEN1KMT2A
SCHEMBL2591063 0.80 NPY5R (1.00) NPY5RABCG2MEN1KMT2APDE5A
SCHEMBL10135169 0.79 CSNK2A1 (0.59) CSNK2A1ABCG2MEN1KMT2AEGFR
SCHEMBL4972017 0.79 CSNK2A1 (1.00) CSNK2A1CLK4DAPK3PIM1CSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8168651-B2 Protein kinase modulators CYLENE PHARMACEUTICALS, INC. (US) 2012-05-01 US disclosed
US-8168651-B2 Protein kinase modulators CYLENE PHARMACEUTICALS, INC. (US) 2012-05-01 US disclosed