SCHEMBL1014074

SCHEMBL1014074

CC(=O)Nc1ccc(CO)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.61
L3MBTL1 Q9Y468 2/20 0.61
HTT P42858 1/20 0.61
TSHR P16473 2/20 0.59
KMT2A Q03164 6/20 0.59
ALDH1A1 P00352 4/20 0.59
MEN1 O00255 4/20 0.59
MAPT P10636 3/20 0.59
TDP1 Q9NUW8 2/20 0.59
CA12 O43570 1/20 0.59
BRD4 O60885 1/20 0.59
NR1I2 O75469 1/20 0.59
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
MB P02144 1/20 0.59
CYP1A1 P04798 1/20 0.59
CA3 P07451 1/20 0.59
CYP3A4 P08684 1/20 0.59
RARG P13631 1/20 0.59
ALOX5AP P20292 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5464759 0.94 MAPT (0.63) SMN1; SMN2L3MBTL1HTTTSHRKMT2A
SCHEMBL15807633 0.85 MAPT (0.69) L3MBTL1HTTKMT2AALDH1A1MEN1
SCHEMBL274924 0.84 TSHR (0.79) SMN1; SMN2L3MBTL1HTTTSHRKMT2A
SCHEMBL29622963 0.84 AOC3 (0.67) SMN1; SMN2L3MBTL1HTTTSHRKMT2A
SCHEMBL29622962 0.84 AOC3 (0.67) SMN1; SMN2L3MBTL1HTTTSHRKMT2A
SCHEMBL5442187 0.83 FYN (0.45) SMN1; SMN2L3MBTL1HTTTSHRKMT2A
SCHEMBL861674 0.83 SMN1; SMN2 (0.84) SMN1; SMN2L3MBTL1HTTTSHRKMT2A
SCHEMBL6629816 0.83 SMN1; SMN2 (0.57) SMN1; SMN2L3MBTL1HTTTSHRKMT2A
SCHEMBL839533 0.83 SMN1; SMN2 (0.61) SMN1; SMN2L3MBTL1HTTTSHRKMT2A
SCHEMBL155297 0.83 RAB9A (0.64) SMN1; SMN2L3MBTL1HTTTSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 143 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10584213-B2 Phosphazene-containing polyhexahydrotriazine elastomers INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2020-03-10 US claimed
US-20200048417-A1 PHOSPHAZENE-CONTAINING POLYHEXAHYDROTRIAZINE ELASTOMERS INTERNATIONAL BUSINESS MACHINES CORPORATION 2020-02-13 US claimed
US-20240318325-A1 ELECTROCHEMICAL HYDROGENOLYSIS OF CARBONYL GROUPS IN ALDEHYDES AND KETONES USING ZINC CATHODES WISCONSIN ALUMNI RESEARCH FOUNDATION 2024-09-26 US disclosed
WO-2024196478-A1 ELECTROCHEMICAL HYDROGENOLYSIS OF CARBONYL GROUPS IN ALDEHYDES AND KETONES USING ZINC CATHODES WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2024-09-26 WO disclosed
CN-113462278-B Varnish composition, method for producing polyimide resin, and additive 东京应化工业株式会社 2024-06-07 CN disclosed
WO-2023066314-A1 BICYCLIC PEPTIDE LIGAND FOR NECTIN-4 AND USE THEREOF 海思科医药集团股份有限公司 2023-04-27 WO disclosed
CN-114436767-A Method for preparing alcohol compound based on carbonyl reduction catalyzed by zinc acetate 延安大学 2022-05-06 CN disclosed
CN-113474156-B Polyamic acid resin composition, polyimide resin film and method for producing same, laminate, and electronic device and method for producing same 东丽株式会社 2022-04-29 CN disclosed
CN-110312719-B Imidazopyrrolopyridines as JAK family kinase inhibitors 詹森药业有限公司 2022-04-15 CN disclosed
CN-113474156-A Polyamic acid resin composition, polyimide resin film and method for producing same, laminate, and electronic device and method for producing same 东丽株式会社 2021-10-01 CN disclosed
EP-3475262-B1 BICYCLIC IMIDAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF RENAL DISEASE, CARDIOVASCULAR DISEASES AND FIBROTIC DISORDERS BOEHRINGER INGELHEIM INT (DE) 2021-03-24 EP disclosed
EP-0659181-A1 SULFONAMIDE INHIBITORS OF HIV-ASPARTYL PROTEASE VERTEX PHARMACEUTICALS INCORPORATED (US) 1995-06-28 EP disclosed
WO-1995009159-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1995-04-06 WO disclosed
US-5399566-A Hypotensive MEIJI SEIKA KABUSHIKI KAISHA (JP) 1995-03-21 US disclosed
WO-1994005639-A1 SULFONAMIDE INHIBITORS OF HIV-ASPARTYL PROTEASE VERTEX PHARMACEUTICALS INCORPORATED (US) 1994-03-17 WO disclosed
EP-0487745-A1 PYRIDINE DERIVATIVE WITH ANGIOTENSIN II ANTAGONISM MEIJI SEIKA KABUSHIKI KAISHA (JP) 1992-06-03 EP disclosed
EP-0100158-A2 (3-pyridinyl)heteroalkarylalkanols, alkanoic acids and esters THE UPJOHN COMPANY (US) 1984-02-08 EP disclosed
EP-0034752-B1 PHENOXYALKANE DERIVATIVE AND PROCESSES FOR PREPARING SAME Tanabe Seiyaku Co., Ltd. (JP) 1983-06-08 EP disclosed
US-4332809-A ANTIALLERGENS TANABE SEIYAKU CO., LTD. (JP) 1982-06-01 US disclosed
EP-0034752-A1 Phenoxyalkane derivative and processes for preparing same Tanabe Seiyaku Co., Ltd. (JP) 1981-09-02 EP disclosed