SCHEMBL10145979

SCHEMBL10145979

Cn1c(=O)n(CC(C)(C)C)c2ccc(-c3cnccc3N)cc21

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 17/20 0.58
PARG Q86W56 1/20 0.42
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
CYP2C19 P33261 1/20 0.40
PTAFR P25105 1/20 0.38
HTR2B P41595 1/20 0.38
METAP2 P50579 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10146342 0.91 GRM2 (0.47) GRM2PARGCYP1A2CYP3A4CYP2D6
SCHEMBL10146344 0.90 METAP2 (0.48) GRM2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL14992426 0.84 GRM2 (0.56) GRM2PARGPTAFRHTR2B
SCHEMBL14993200 0.84 GRM2 (0.56) GRM2PARGPTAFRHTR2B
SCHEMBL14992658 0.84 GRM2 (0.58) GRM2PARGMETAP2
SCHEMBL10146668 0.83 GRM2 (0.70) GRM2PARGMETAP2
SCHEMBL10146655 0.83 GRM2 (0.48) GRM2PARGCYP1A2CYP3A4CYP2D6
SCHEMBL10145981 0.83 CYP11B1 (0.39) GRM2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL10146361 0.82 GRM2 (0.62) GRM2PARGPTAFRHTR2B
SCHEMBL14992270 0.82 GRM2 (0.56) GRM2PARGPTAFRHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021382-A1 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2012-02-16 WO disclosed