SCHEMBL10146342

SCHEMBL10146342

Cn1c(=O)n(CC(C)(C)F)c2ccc(-c3cnccc3N)cc21

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 3/20 0.47
METAP2 P50579 3/20 0.41
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
CYP2C19 P33261 1/20 0.39
GRIN1 Q05586 10/20 0.36
GRIN2B Q13224 10/20 0.36
MAPK14 Q16539 1/20 0.35
BCL6 P41182 1/20 0.35
PARG Q86W56 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10146344 0.92 METAP2 (0.48) GRM2METAP2CYP1A2CYP3A4CYP2D6
SCHEMBL10145979 0.91 GRM2 (0.58) GRM2METAP2CYP1A2CYP3A4CYP2D6
SCHEMBL14992455 0.85 GRM2 (0.46) GRM2METAP2GRIN1GRIN2BBCL6
SCHEMBL10145981 0.81 CYP11B1 (0.39) GRM2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL14992426 0.80 GRM2 (0.56) GRM2GRIN1GRIN2BPARG
SCHEMBL10146644 0.80 GRM2 (0.52) GRM2CYP11B2GRIN1GRIN2B
SCHEMBL14992270 0.78 GRM2 (0.56) GRM2GRIN1GRIN2BPARG
SCHEMBL14992658 0.78 GRM2 (0.58) GRM2METAP2GRIN1GRIN2BPARG
SCHEMBL14992498 0.77 GRM2 (0.44) GRM2METAP2GRIN1GRIN2B
SCHEMBL14993200 0.76 GRM2 (0.56) GRM2PARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021382-A1 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2012-02-16 WO disclosed