SCHEMBL10146161

SCHEMBL10146161

C=S1(=O)CCN(C(=O)c2cnc(N3CCC(C)(C)c4ccccc43)nc2C(F)(F)F)CC1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RY1 P47900 2/20 0.37
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
OPRL1 P41146 2/20 0.35
HCRTR1 O43613 3/20 0.33
HCRTR2 O43614 3/20 0.33
PDE4B Q07343 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
NR1H2 P55055 3/20 0.33
PDK2 Q15119 1/20 0.33
JUN P05412 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
CXCR4 P61073 1/20 0.32
HSD11B1 P28845 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL541322 0.93 OPRL1 (0.41) P2RY1RXRARXRBRXRGOPRL1
SCHEMBL541323 0.91 P2RY1 (0.38) P2RY1RXRARXRBRXRGOPRL1
SCHEMBL6523323 0.87 PDE4B (0.44) P2RY1OPRL1PDE4BKDM4EALDH1A1
SCHEMBL12796019 0.83 RXRA (0.43) P2RY1RXRARXRBRXRGOPRL1
SCHEMBL12795984 0.81 ALDH1A1 (0.50) P2RY1RXRARXRBRXRGHCRTR1
SCHEMBL12796505 0.69 TSHR (0.48) KDM4EALDH1A1NR1H2NFKB1NFKB2
SCHEMBL12796342 0.68 AVPR1A (0.46) OPRL1
SCHEMBL10145795 0.68 NR1H2 (0.43) P2RY1OPRL1KDM4EALDH1A1NR1H2
SCHEMBL12796228 0.67 NR1H2 (0.43) OPRL1KDM4EALDH1A1NR1H2NFKB1
SCHEMBL12796510 0.67 NR1H2 (0.45) P2RY1RXRARXRBRXRGOPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415765-A1 PYRIMIDINE COMPOUND Astellas Pharma Inc. (JP) 2012-02-08 EP disclosed