SCHEMBL10146396

SCHEMBL10146396

Cc1nc2ncc(C(F)(F)F)cc2[nH]1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 3/20 0.58
SMN1; SMN2 Q16637 2/20 0.57
HSD17B10 Q99714 2/20 0.46
HTT P42858 1/20 0.46
MAPT P10636 2/20 0.44
GAA P10253 1/20 0.44
KDM4E B2RXH2 2/20 0.42
POLB P06746 1/20 0.42
HPGD P15428 1/20 0.42
METAP2 P50579 1/20 0.41
AGBL2 Q5U5Z8 1/20 0.37
RAB9A P51151 1/20 0.37
NPBWR1 P48145 1/20 0.37
BRD4 O60885 1/20 0.36
KCNH2 Q12809 2/20 0.36
PDE2A O00408 2/20 0.36
DGAT1 O75907 1/20 0.35
ADORA2A P29274 1/20 0.35
AURKB Q96GD4 1/20 0.35
TRPA1 O75762 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11773659 0.81 HSD17B10 (0.70) AURKASMN1; SMN2HSD17B10HTTMAPT
SCHEMBL2419692 0.79 HTT (0.54) AURKASMN1; SMN2HSD17B10HTTMAPT
SCHEMBL21263259 0.77 SMN1; SMN2 (0.62) AURKASMN1; SMN2HSD17B10HTTMAPT
SCHEMBL2756735 0.76 SMN1; SMN2 (0.67) AURKASMN1; SMN2HSD17B10HTTMAPT
SCHEMBL29954536 0.76 AURKA (0.48) AURKASMN1; SMN2HSD17B10HTTKDM4E
SCHEMBL20909800 0.74 SMN1; SMN2 (0.65) AURKASMN1; SMN2HSD17B10HTTPOLB
SCHEMBL16739826 0.73 SMN1; SMN2 (0.62) AURKASMN1; SMN2HSD17B10HTTMAPT
SCHEMBL618430 0.73 SMN1; SMN2 (1.00) AURKASMN1; SMN2HTTMAPTKDM4E
SCHEMBL12335638 0.72 POLB (0.42) AURKASMN1; SMN2HSD17B10MAPTGAA
SCHEMBL8265307 0.71 MAPT (0.50) HSD17B10HTTMAPTGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012009217-A1 SPIROCYCLIC COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed