SCHEMBL29954536

SCHEMBL29954536

O=Cc1nc2ncc(C(F)(F)F)cc2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.48
HTT P42858 1/20 0.43
HSD17B10 Q99714 1/20 0.43
METAP2 P50579 1/20 0.38
KCNH2 Q12809 3/20 0.37
DGAT1 O75907 2/20 0.37
ADORA2A P29274 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 1/20 0.35
RAB9A P51151 1/20 0.35
JUN P05412 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
AURKB Q96GD4 1/20 0.33
IDO1 P14902 2/20 0.33
LMNA P02545 1/20 0.33
KMT2A Q03164 1/20 0.33
TRPA1 O75762 1/20 0.33
PDE10A Q9Y233 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11773659 0.77 HSD17B10 (0.70) AURKAHTTHSD17B10METAP2KCNH2
SCHEMBL2419692 0.76 HTT (0.54) AURKAHTTHSD17B10METAP2KCNH2
SCHEMBL10146396 0.76 AURKA (0.58) AURKAHTTHSD17B10METAP2KCNH2
SCHEMBL29951206 0.73 NPBWR1 (0.54) HSD17B10KCNH2DGAT1
SCHEMBL12353892 0.71 CBFB (0.50) HTTJUNNFKB1NFKB2RELA
SCHEMBL23782321 0.70 NPBWR1 (0.40) METAP2KCNH2DGAT1KDM4EKMT2A
SCHEMBL26039481 0.70 IDO1 (0.47) AURKAHTTHSD17B10METAP2KCNH2
SCHEMBL2004991 0.68 METAP2 (0.44) METAP2
SCHEMBL22481479 0.66 DGAT1 (0.43) AURKAKCNH2DGAT1
SCHEMBL10719652 0.66 AURKA (0.41) AURKAHTTHSD17B10METAP2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed