SCHEMBL1014661

SCHEMBL1014661

CC(C)CC(C=O)NC(=O)C(CC(C)C)NC(=O)OCc1ccccc1

nearest known ligand 0.78

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PSMB1 P20618 1/20 0.78
PSMB5 P28074 1/20 0.78
PSMB2 P49721 1/20 0.78
CTSL P07711 11/20 0.73
CTSB P07858 7/20 0.73
CTSK P43235 6/20 0.70
CTSS P25774 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8971981 1.00 PSMB1 (0.78) PSMB1PSMB5PSMB2CTSLCTSB
SCHEMBL3054703 1.00 PSMB1 (0.78) PSMB1PSMB5PSMB2CTSLCTSB
SCHEMBL7710728 1.00 PSMB1 (0.78) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL7862424 0.99 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL14579851 0.99 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL5062219 0.99 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL14514061 0.99 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL13436259 0.99 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL2522088 0.99 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL2535252 0.99 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115551512-A Use of compounds or compositions comprising NLRP1 inflammatory body activation inhibitors for the treatment of airway inflammation in humans 南洋理工大学 2022-12-30 CN claimed
CN-113272294-A 2, 6-bis (((1H-benzo [ D ] imidazol-2-yl) thio) methyl) pyridine and N2, N6-dibenzylpyridine-2, 6-dicarboxamide derivatives and related compounds as phosphoinositide 3-kinase (PI3K) inhibitors for the treatment of cancer 雅典学院生物医学研究基金会 2021-08-17 CN claimed
CN-118215461-A Compositions and methods for reducing pigmentation 总医院公司 2024-06-18 CN disclosed
CN-117355333-A Combination comprising anti-TM 4SF1 antibody and immunotherapeutic agent and method of use thereof 安吉克公司 2024-01-05 CN disclosed
CN-115551512-A Use of compounds or compositions comprising NLRP1 inflammatory body activation inhibitors for the treatment of airway inflammation in humans 南洋理工大学 2022-12-30 CN disclosed
CN-113272294-A 2, 6-bis (((1H-benzo [ D ] imidazol-2-yl) thio) methyl) pyridine and N2, N6-dibenzylpyridine-2, 6-dicarboxamide derivatives and related compounds as phosphoinositide 3-kinase (PI3K) inhibitors for the treatment of cancer 雅典学院生物医学研究基金会 2021-08-17 CN disclosed
CN-112359018-A Methods and compositions for regenerating hair cells and/or supporting cells 麻省眼耳医院 2021-02-12 CN disclosed
CN-105641700-B Means and methods for combating muscle disorders 莱顿教学医院 2021-01-01 CN disclosed
CN-104869987-B Methods and compositions for regenerating hair cells and/or supporting cells 麻省眼耳医院 2020-10-16 CN disclosed
US-9128081-B2 TDP-43-storing cell model TOKYO METROPOLITAN INSTITUTE OF MEDICAL SCIENCE (JP) 2015-09-08 US disclosed
EP-2272955-B1 TDP-43-STORING CELL MODEL TOKYO METROPOLITAN INST MEDICAL SCIENCE (JP) 2015-08-26 EP disclosed
US-8715643-B2 TDP-43-storing cell model TOKYO METROPOLITAN INSTITUTE OF MEDICAL SCIENCE (JP) 2014-05-06 US disclosed
US-20140099660-A1 TDP-43-STORING CELL MODEL TOKYO METROPOLITIAN INSTITUTE OF MEDICAL SCIENCE (JP) 2014-04-10 US disclosed
US-20110034447-A1 TDP-43-STORING CELL MODEL TOKYO METROPOLITAN INSTITUTE OF MEDICAL SCIENCE (JP) 2011-02-10 US disclosed
EP-2272955-A1 TDP-43-STORING CELL MODEL Tokyo Metropolitan Organization for Medical Research (JP) 2011-01-12 EP disclosed