SCHEMBL10147580

SCHEMBL10147580

Cn1nc(C(C)(C)C)cc1-c1nnc(C(C)(C)[S+]([O-])Cc2ccc(F)cc2)o1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP1A2 P05177 1/20 0.30
GALR3 O60755 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL352485 0.80 ALDH1A1 (0.35) ALDH1A1MAPTMAPK1NPSR1CYP1A2
SCHEMBL10147582 0.79
SCHEMBL351008 0.77 CNR2 (0.39) CYP1A2RAB9A
SCHEMBL10147588 0.75 CYP1A2 (0.33) CYP1A2RAB9A
SCHEMBL10146105 0.74 CYP1A2 (0.44) CYP1A2
SCHEMBL13618724 0.71 GRN (0.40) CYP1A2
SCHEMBL350907 0.66 CNR2 (0.51) ALDH1A1MAPTRAB9A
SCHEMBL10147542 0.65 MAPK13 (0.37) MAPT
SCHEMBL350932 0.61 ALDH1A1 (0.35) ALDH1A1MAPTMAPK1NPSR1
SCHEMBL351826 0.61 CNR2 (0.36) ALDH1A1NPSR1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2418207-A1 Sulfone compounds which modulate the CB2 receptor Boehringer Ingelheim International GmbH (DE) 2012-02-15 EP disclosed