SCHEMBL10151395

SCHEMBL10151395

COc1ccc2c(c1)nc(C(F)(F)F)n2-c1cnc(NC(=O)c2cc(I)ccc2OC)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.41
NPC1 O15118 5/20 0.41
MITF O75030 1/20 0.41
TP53 P04637 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 6/20 0.38
RXFP1 Q9HBX9 2/20 0.38
MAPT P10636 2/20 0.38
CACNA1D Q01668 1/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MEN1 O00255 4/20 0.36
HPGDS O60760 1/20 0.36
ABCB1 P08183 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HCRTR1 O43613 1/20 0.35
BRD4 O60885 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL645446 0.91 ABCB1 (0.44) RAB9ANPC1MITFTP53GAA
SCHEMBL645416 0.90 NPC1 (0.44) RAB9ANPC1MITFTP53GAA
SCHEMBL14400700 0.90 RAB9A (0.39) RAB9ANPC1MITFTP53GAA
SCHEMBL648285 0.89 KMT2A (0.46) RAB9ANPC1MITFTP53GAA
SCHEMBL649492 0.89 NPC1 (0.51) RAB9ANPC1MITFTP53GAA
SCHEMBL645754 0.87 HPGDS (0.40) RAB9ANPC1MITFTP53GAA
SCHEMBL647532 0.86 NPC1 (0.41) RAB9ANPC1TP53GAAKMT2A
SCHEMBL8234095 0.86 NPC1 (0.55) RAB9ANPC1MITFTP53GAA
SCHEMBL645960 0.86 NPC1 (0.46) RAB9ANPC1MITFTP53GAA
SCHEMBL646333 0.86 NPC1 (0.46) RAB9ANPC1TP53GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119643-B2 Benzoimidazolyl-pyrazine compounds for inflammation and immune-related uses SYNTA PHARMACEUTICALS CORP. (US) 2012-02-21 US disclosed