SCHEMBL10151560

SCHEMBL10151560

CC(C)(C)OC(=O)N1CCN(C(=O)NC[C@H]2CN(c3ccc(N4CCN(C(=O)OCc5ccccc5)N(C(=O)OCc5ccccc5)CC4)c(F)c3)C(=O)O2)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOB P27338 7/20 0.54
MAOA P21397 4/20 0.54
LMNA P02545 1/20 0.52
PTGS1 P23219 1/20 0.52
CALML3 P27482 1/20 0.52
SDHA P31040 1/20 0.52
F10 P00742 12/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15827739 0.95 MAOB (0.49) MAOBMAOALMNAPTGS1CALML3
SCHEMBL10151452 0.93 MAOB (0.62) MAOBMAOALMNAPTGS1CALML3
SCHEMBL10151562 0.89 MAOB (0.51) MAOBMAOALMNAPTGS1CALML3
SCHEMBL10151456 0.89 MAOB (0.49) MAOBMAOALMNAPTGS1CALML3
SCHEMBL5725608 0.88 MAOB (0.56) MAOBMAOALMNAPTGS1CALML3
SCHEMBL5725604 0.88 MAOB (0.56) MAOBMAOALMNAPTGS1CALML3
SCHEMBL10151454 0.88 MAOB (0.48) MAOBMAOALMNAPTGS1CALML3
SCHEMBL10151523 0.87 MAOB (0.53) MAOBMAOALMNAPTGS1CALML3
SCHEMBL13357833 0.86 MAOB (0.46) MAOBMAOALMNAPTGS1CALML3
SCHEMBL5323788 0.85 MAOB (0.67) MAOBMAOALMNAPTGS1CALML3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8785625-B2 Compound having heterocyclic ring RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2014-07-22 US disclosed
US-20120208997-A1 NOVEL COMPOUND HAVING HETEROCYCLIC RING SUZUKI HIDEYUKI (JP) 2012-08-16 US disclosed
US-20120208997-A1 NOVEL COMPOUND HAVING HETEROCYCLIC RING SUZUKI HIDEYUKI (JP) 2012-08-16 US disclosed
US-8148362-B2 Compound having heterocyclic ring RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2012-04-03 US disclosed
US-8148362-B2 Compound having heterocyclic ring RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2012-04-03 US disclosed
US-20090299059-A1 Novel Compound Having Heterocyclic Ring RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2009-12-03 US disclosed
US-20090299059-A1 Novel Compound Having Heterocyclic Ring RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2009-12-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090299059-A1 Novel Compound Having Heterocyclic Ring NR0B2, NR2C2, NR0B1 MAOB 2611/4885MAOA 2965/4885LMNA 4493/4885
US-20120208997-A1 NOVEL COMPOUND HAVING HETEROCYCLIC RING OXA1L, MRPL21, TOP1 MAOB 1404/4885MAOA 1563/4885LMNA 3275/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.