SCHEMBL10153699

SCHEMBL10153699

O=C(NC1CCCC1)C1C(=O)N(O)C(=O)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 7/20 0.57
HTT P42858 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
GAA P10253 1/20 0.52
TP53 P04637 1/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
RECQL P46063 1/20 0.49
NPSR1 Q6W5P4 1/20 0.48
MCHR1 Q99705 1/20 0.48
MAPT P10636 1/20 0.48
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
THRB P10828 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31653964 0.99 TSHR (0.59) TSHRHTTL3MBTL1GAATP53
SCHEMBL9958705 0.80 HDAC4 (0.62) TSHRHTTL3MBTL1GAAALDH1A1
SCHEMBL19380274 0.79 HDAC4 (0.44) TSHRHTTL3MBTL1GAAALDH1A1
SCHEMBL10154010 0.78 MAPT (0.44) TSHRHTTL3MBTL1MAPTTHRB
SCHEMBL9958546 0.78 TSHR (0.48) TSHRHTTL3MBTL1GAATP53
SCHEMBL31653962 0.77 MEN1 (0.47) L3MBTL1GAALMNANPSR1
SCHEMBL10153609 0.77 MEN1 (0.47) L3MBTL1GAALMNANPSR1
SCHEMBL10153606 0.76 KCNA5 (0.48) L3MBTL1GAALMNAMAPT
SCHEMBL31653994 0.76 KCNA5 (0.48) L3MBTL1GAALMNAMAPT
SCHEMBL11789850 0.75 ALDH1A1 (0.43) HTTGAAALDH1A1LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed