SCHEMBL10155702

SCHEMBL10155702

NCC1(c2cccc([N+](=O)[O-])c2)CCCC1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 11/20 0.55
SLC6A4 P31645 10/20 0.55
DPP4 P27487 1/20 0.53
KDM1A O60341 1/20 0.52
SLC6A2 P23975 4/20 0.48
LMNA P02545 2/20 0.47
TSHR P16473 1/20 0.47
ALDH1A1 P00352 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10669384 0.86 KDM1A (0.48) SLC6A3SLC6A4KDM1ALMNATSHR
SCHEMBL10155679 0.80 KDM1A (0.56) KDM1ALMNATSHRALDH1A1
SCHEMBL28218216 0.78 KDM1A (0.55) SLC6A3KDM1ASLC6A2LMNATSHR
SCHEMBL26218870 0.78 KDM1A (0.54) SLC6A3KDM1ASLC6A2LMNATSHR
SCHEMBL26218874 0.76 KDM1A (0.53) SLC6A3KDM1ASLC6A2LMNATSHR
SCHEMBL2817503 0.74 MAOA (0.52) SLC6A3SLC6A4DPP4SLC6A2TSHR
SCHEMBL10184986 0.74 TSHR (0.57) SLC6A3KDM1ASLC6A2LMNATSHR
SCHEMBL30492221 0.74 KDM1A (0.50) KDM1ALMNATSHRALDH1A1TDP1
SCHEMBL6676866 0.73 AKR1C1 (0.57) KDM1ALMNATSHRALDH1A1
SCHEMBL2814607 0.73 KDM1A (0.49) SLC6A3KDM1ASLC6A2LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120015961-A1 ISOTHIOUREA DERIVATIVES OR ISOUREA DERIVATIVES HAVING BACE1 INHIBITORY ACTIVITY SHIONOGI & CO., LTD. (JP) 2012-01-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120015961-A1 ISOTHIOUREA DERIVATIVES OR ISOUREA DERIVATIVES HAVING BACE1 INHIBITORY ACTIVITY BACE1, BACE2, APP SLC6A3 322/4885SLC6A4 912/4885DPP4 79/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.