SCHEMBL10157014

SCHEMBL10157014

N#Cc1cc(COc2ccccc2)ccn1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.56
CYP11B1 P15538 2/20 0.44
CYP11B2 P19099 1/20 0.44
FFAR1 O14842 2/20 0.44
FFAR4 Q5NUL3 1/20 0.44
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
LMNA P02545 1/20 0.43
PTGS1 P23219 1/20 0.43
SLC6A2 P23975 1/20 0.43
PTGS2 P35354 1/20 0.43
SLC6A3 Q01959 1/20 0.43
HIF1A Q16665 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
GRM5 P41594 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
APP P05067 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
MAOA P21397 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12439723 0.84 MAOB (0.62) MAOBCYP1A2CYP2C19LMNAPTGS1
SCHEMBL20385730 0.80 NOS3 (0.44) MAOBCYP11B1CYP11B2GRM5MAOA
SCHEMBL1145726 0.78 GRM5 (0.39) MAOBCYP11B1CYP11B2GRM5
SCHEMBL6479355 0.78 CALM1 (0.43) MAOBCYP1A2CYP2C19LMNACYP3A4
SCHEMBL1145730 0.78 GRM5 (0.41) GRM5MAOAALDH1A1
SCHEMBL4016988 0.75 GRM5 (0.38) GRM5
SCHEMBL25909279 0.75 MAOB (0.42) MAOBCYP11B1CYP11B2GRM5MAOA
SCHEMBL1248693 0.75 MAOB (0.66) MAOBFFAR1FFAR4GRM5MAOA
SCHEMBL10157091 0.75 GRM5 (0.49) MAOBFFAR1CYP1A2CYP2C19LMNA
SCHEMBL3370181 0.75 GRM5 (0.52) MAOBCYP11B1CYP11B2CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012052390-A1 N-2-(2-PYRIDINYL)-4-PYRIMIDINYL-BETA-ALANINE DERIVATIVES AS INHIBITORS OF HISTONE DEMETHYLASE JMJD3 GLAXO GROUP LIMITED (GB) 2012-04-26 WO disclosed