SCHEMBL10157720

SCHEMBL10157720

O=C(CO)c1cc(OCc2ccccc2)no1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 3/20 0.59
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
NR4A2 P43354 2/20 0.40
PTGES O14684 1/20 0.40
ALOX5 P09917 1/20 0.40
KDM5A P29375 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
FOLH1 Q04609 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
NR4A1 P22736 1/20 0.40
NR4A3 Q92570 1/20 0.40
GABRA5 P31644 1/20 0.39
P4HTM Q9NXG6 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10524070 0.87 SMPD1 (0.57) SMPD1MEN1KMT2ANR4A2PTGES
SCHEMBL630848 0.86 SMPD1 (0.63) SMPD1MEN1KMT2ANR4A2PTGES
SCHEMBL10521252 0.84 SMPD1 (0.60) SMPD1MEN1KMT2APTGESALOX5
SCHEMBL10519525 0.84 SMPD1 (0.60) SMPD1MEN1KMT2ANR4A2PTGES
SCHEMBL12909761 0.81 SMPD1 (0.57) SMPD1MEN1KMT2ANR4A2PTGES
SCHEMBL630644 0.81 SMPD1 (0.61) SMPD1MEN1KMT2APTGESALOX5
SCHEMBL12568619 0.80 SMPD1 (0.56) SMPD1MEN1KMT2ANR4A2PTGES
SCHEMBL15004563 0.80 SMPD1 (0.67) SMPD1MEN1KMT2APTGESALOX5
SCHEMBL322866 0.78 SMPD1 (0.53) SMPD1NPC1RAB9A
SCHEMBL22777760 0.78 SMPD1 (0.76) SMPD1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8907104-B2 Synthesis of enone intermediate PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2014-12-09 US disclosed
US-20140179929-A1 SYNTHESIS OF ENONE INTERMEDIATE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2014-06-26 US disclosed
US-8580969-B2 Synthesis of enone intermediate PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2013-11-12 US disclosed
US-20130217886-A1 SYNTHESIS OF ENONE INTERMEDIATE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2013-08-22 US disclosed
US-8293920-B2 Synthesis of enone intermediate PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-10-23 US disclosed
US-20120029199-A1 SYNTHESIS OF ENONE INTERMEDIATE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-02-02 US disclosed
US-7960559-B2 Synthesis of enone intermediate PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2011-06-14 US disclosed
US-20110009639-A1 SYNTHESIS OF ENONE INTERMEDIATE MYERS ANDREW G 2011-01-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130217886-A1 SYNTHESIS OF ENONE INTERMEDIATE TECR, ECI1, ERAL1 SMPD1 4418/4885MEN1 608/4885KMT2A 3374/4885
US-20110009639-A1 SYNTHESIS OF ENONE INTERMEDIATE TECR, ECI1, ERAL1 SMPD1 4418/4885MEN1 608/4885KMT2A 3374/4885
US-20140179929-A1 SYNTHESIS OF ENONE INTERMEDIATE TECR, ECI1, ERAL1 SMPD1 4418/4885MEN1 608/4885KMT2A 3374/4885
US-20120029199-A1 SYNTHESIS OF ENONE INTERMEDIATE TECR, ECI1, ERAL1 SMPD1 4418/4885MEN1 608/4885KMT2A 3374/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.