SCHEMBL10163519

SCHEMBL10163519

COc1ccccc1CNC(=O)C=O

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.63
KMT2A Q03164 4/20 0.60
MEN1 O00255 3/20 0.60
ALDH1A1 P00352 3/20 0.60
HTT P42858 2/20 0.60
NPC1 O15118 2/20 0.60
RAB9A P51151 2/20 0.60
NPSR1 Q6W5P4 1/20 0.60
HDAC1 Q13547 1/20 0.58
POLB P06746 1/20 0.57
MAPT P10636 1/20 0.57
BLM P54132 1/20 0.57
GAA P10253 1/20 0.57
KDM4E B2RXH2 1/20 0.57
RCE1 Q9Y256 1/20 0.57
TSHR P16473 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8765637 0.86 HPGD (0.61) HPGDKMT2AMEN1ALDH1A1HTT
SCHEMBL885000 0.81 MTNR1A (0.71) HPGDKMT2AMEN1ALDH1A1HTT
SCHEMBL13434069 0.81 HPGD (0.69) HPGDKMT2AMEN1ALDH1A1HTT
SCHEMBL2938380 0.81 KMT2A (0.69) HPGDKMT2AMEN1ALDH1A1HTT
SCHEMBL14667212 0.81 KMT2A (0.65) HPGDKMT2AMEN1ALDH1A1HTT
SCHEMBL18971048 0.80 APLNR (0.64) HPGDKMT2AMEN1ALDH1A1HTT
SCHEMBL15338437 0.80 HDAC3 (0.50) HDAC1
SCHEMBL1520822 0.80 NPSR1 (0.68) HPGDKMT2AMEN1ALDH1A1HTT
SCHEMBL10163441 0.79 HPGD (0.65) HPGDKMT2AMEN1ALDH1A1HTT
SCHEMBL14670856 0.79 HPGD (0.70) HPGDKMT2AMEN1ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2409985-A2 Inhibitors de serine proteases, especially of the NS3 protease of the hepatitis C virus VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-01-25 EP disclosed