SCHEMBL10167993

SCHEMBL10167993

[C-]#[N+]c1ccnc(N2CCN(C(=O)OCC(C)(C)C)CC2)c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
OPRD1 P41143 1/20 0.41
KCNH2 Q12809 1/20 0.41
SMO Q99835 1/20 0.41
IDE P14735 1/20 0.40
HRH3 Q9Y5N1 7/20 0.39
PIK3CA P42336 1/20 0.38
HTT P42858 1/20 0.38
NOS1 P29475 2/20 0.38
NOS2 P35228 2/20 0.38
LRRK2 Q5S007 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NOS3 P29474 1/20 0.37
GPR119 Q8TDV5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL390651 0.85 NOS1 (0.49) HPGDSMN1; SMN2OPRD1KCNH2SMO
SCHEMBL390540 0.84 OPRD1 (0.57) HPGDSMN1; SMN2OPRD1KCNH2SMO
SCHEMBL390619 0.83 HRH3 (0.56) HPGDSMN1; SMN2OPRD1KCNH2SMO
SCHEMBL390340 0.83 HRH3 (0.54) HPGDSMN1; SMN2OPRD1KCNH2SMO
SCHEMBL10168032 0.82 HSD17B10 (0.44) HPGDSMN1; SMN2SMONPSR1
SCHEMBL388016 0.82 HRH3 (0.57) HPGDSMN1; SMN2KCNH2HRH3
SCHEMBL389756 0.81 HRH3 (0.56) HPGDSMN1; SMN2OPRD1KCNH2SMO
SCHEMBL390338 0.81 HRH3 (0.56) HPGDSMN1; SMN2OPRD1KCNH2SMO
SCHEMBL14340961 0.81 MAPT (0.49) HPGDSMN1; SMN2OPRD1KCNH2SMO
SCHEMBL388764 0.81 GRIN2D (0.49) HPGDSMN1; SMN2OPRD1KCNH2SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8101618-B2 1,4-substituted piperazine derivatives MSD K.K. (JP) 2012-01-24 US disclosed
US-20090062293-A1 1,4-Substituted Piperazine Derivatives MSD K.K. (JP) 2009-03-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090062293-A1 1,4-Substituted Piperazine Derivatives GRIN1, GRM1, GRIN2C HPGD 2246/4885SMN1; SMN2 960/4885OPRD1 37/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.