SCHEMBL10168575

SCHEMBL10168575

CC(C)N1CCCC2(CC(c3ccncc3)=NO2)C1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
PKM P14618 1/20 0.34
ABL1 P00519 1/20 0.34
RIN1 Q13671 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
SSTR5 P35346 3/20 0.34
USP2 O75604 1/20 0.32
CYP3A4 P08684 2/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10168605 0.89 CHRNB4 (0.52) CHRNB4CHRNA3SSTR5CYP1A2CYP2D6
SCHEMBL10168595 0.86 CRBN (0.42) CHRNB4CHRNA3USP2CYP1A2
SCHEMBL10210779 0.83 CHRNB4 (0.42) CHRNB4CHRNA3PKMABL1RIN1
SCHEMBL10168587 0.80 PYGL (0.39) CHRNB4CHRNA3PKMSSTR5
SCHEMBL10168567 0.80 CHRNB4 (0.36) CHRNB4CHRNA3CYP1A2CYP2D6HSD17B10
SCHEMBL10168667 0.76
SCHEMBL10212112 0.75 CRBN (0.40) CHRNB4CHRNA3PKMTDP1SSTR5
SCHEMBL25466551 0.74
SCHEMBL10168596 0.74
SCHEMBL14507947 0.72 CHRNB4 (0.50) CHRNB4CHRNA3SSTR5CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8586751-B2 Nicotinamide compounds useful as kinase modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2013-11-19 US disclosed
US-20120082702-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL-MEYERS SQUIBB COMPANY 2012-04-05 US disclosed
US-20120082702-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL-MEYERS SQUIBB COMPANY 2012-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120082702-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS NADK, BTK, NAMPT CHRNB4 2625/4885CHRNA3 2203/4885PKM 981/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.