SCHEMBL10169503

SCHEMBL10169503

CC(C)c1cccc(NS(=O)(=O)CCCCl)c1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 1/20 0.47
CA2 P00918 1/20 0.41
EGFR P00533 1/20 0.41
TNNI3K Q59H18 1/20 0.41
ALOX12 P18054 1/20 0.39
PGR P06401 1/20 0.39
BRD4 O60885 1/20 0.38
CBLB Q13191 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22220775 0.82 CA2 (0.47) ADRB3CA2EGFRTNNI3KALOX12
SCHEMBL10191948 0.81 HPGD (0.46) ADRB3
SCHEMBL10100499 0.76 KEAP1 (0.55) CA2EGFRTNNI3KBRD4
SCHEMBL6830181 0.76 AR (0.50) CA2PGR
SCHEMBL10876109 0.74 CDK1 (0.52) CA2
SCHEMBL693060 0.74 ADRB3 (0.39) ADRB3BRD4
SCHEMBL14508412 0.73 CA2 (0.55) CA2EGFRTNNI3KALOX12PGR
SCHEMBL13181439 0.73 KDM1A (0.48) ADRB3CA2EGFRTNNI3KALOX12
SCHEMBL27182647 0.72 CA2 (0.50) CA2EGFRTNNI3KALOX12PGR
SCHEMBL10169501 0.71 KDM4E (0.35) CA2EGFRTNNI3KALOX12PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8586751-B2 Nicotinamide compounds useful as kinase modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2013-11-19 US disclosed
US-20120082702-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL-MEYERS SQUIBB COMPANY 2012-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120082702-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS NADK, BTK, NAMPT ADRB3 2669/4885CA2 2566/4885EGFR 2225/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.