SCHEMBL10175112

SCHEMBL10175112

COC(=O)c1ccc2c(c1)nc(-c1cccnc1)n2C

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.64
CYP11B1 P15538 2/20 0.58
CYP11B2 P19099 2/20 0.58
CYP19A1 P11511 1/20 0.58
HDAC1 Q13547 3/20 0.54
HDAC8 Q9BY41 3/20 0.54
HDAC6 Q9UBN7 3/20 0.54
SLC2A1 P11166 1/20 0.52
HDAC3 O15379 2/20 0.51
HDAC2 Q92769 2/20 0.51
KDM4E B2RXH2 2/20 0.49
NR4A2 P43354 1/20 0.49
KIT P10721 2/20 0.48
ALDH1A1 P00352 1/20 0.48
ABL1 P00519 1/20 0.47
BCR P11274 1/20 0.47
SRC P12931 1/20 0.47
MAPT P10636 2/20 0.47
NPC1 O15118 1/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896670 0.87 NAMPT (0.67) NAMPTCYP11B1CYP11B2HDAC1HDAC8
SCHEMBL10175457 0.86 NAMPT (0.70) NAMPTCYP11B1CYP11B2HDAC1HDAC8
SCHEMBL17896668 0.84 NAMPT (0.61) NAMPTCYP11B1CYP11B2HDAC1HDAC8
SCHEMBL17896675 0.84 CYP11B2 (0.63) CYP11B1CYP11B2CYP19A1SLC2A1
SCHEMBL17896669 0.83 HDAC1 (0.50) NAMPTCYP11B1CYP11B2CYP19A1HDAC1
SCHEMBL19763370 0.82 HDAC6 (0.59) NAMPTHDAC1HDAC8HDAC6HDAC3
SCHEMBL10175817 0.79 RAD51 (0.60) NAMPTCYP11B1CYP11B2CYP19A1KDM4E
SCHEMBL10175103 0.79 NAMPT (0.61) NAMPTCYP11B1CYP11B2KITALDH1A1
SCHEMBL7812395 0.78 CYP11B2 (0.58) NAMPTCYP11B1CYP11B2CYP19A1SLC2A1
SCHEMBL30158985 0.78 NPC1 (0.61) NAMPTHDAC1HDAC8HDAC6HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed