SCHEMBL10176220

SCHEMBL10176220

COc1cncc(-c2nc3cc(Cl)c(Cl)cc3n2C2CC2)c1C

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 17/20 0.56
CYP11B1 P15538 16/20 0.56
CYP3A4 P08684 1/20 0.56
CCNT1 O60563 2/20 0.48
CDK9 P50750 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896695 0.86 CYP11B2 (0.55) CYP11B2CYP11B1CYP3A4
SCHEMBL10175802 0.86 CYP11B2 (0.76) CYP11B2CYP11B1CYP3A4
SCHEMBL17896658 0.82 POLB (0.45) CYP11B2CYP11B1CYP3A4CCNT1CDK9
SCHEMBL17896662 0.78 CYP11B2 (0.75) CYP11B2CYP11B1CCNT1CDK9
SCHEMBL10176222 0.75 CYP11B2 (0.60) CYP11B2CYP11B1CYP3A4CCNT1CDK9
SCHEMBL17896663 0.74 CYP11B2 (0.56) CYP11B2CYP11B1CYP3A4CCNT1CDK9
SCHEMBL459367 0.72 CYP11B2 (1.00) CYP11B2CYP11B1CYP3A4
SCHEMBL10176217 0.71 CYP11B2 (0.62) CYP11B2CYP11B1CYP3A4
SCHEMBL17896661 0.71 CYP11B1 (0.86) CYP11B2CYP11B1CCNT1CDK9
SCHEMBL10175800 0.71 CYP11B2 (1.00) CYP11B2CYP11B1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed