SCHEMBL1018100

SCHEMBL1018100

CCCCCc1nc[nH]n1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.36
GPR84 Q9NQS5 2/20 0.36
HCAR2 Q8TDS4 2/20 0.36
HCAR3 P49019 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
PAK1 Q13153 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP3A4 P08684 1/20 0.33
PTGS2 P35354 1/20 0.33
PI4KA P42356 1/20 0.33
PI4K2B Q8TCG2 1/20 0.33
PI4K2A Q9BTU6 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26111611 0.98 KCNH2 (0.39) KCNH2GPR84HCAR2HCAR3CYP3A4
SCHEMBL11444203 0.98 KCNH2 (0.39) KCNH2GPR84HCAR2HCAR3CYP3A4
SCHEMBL26112848 0.98 KCNH2 (0.39) KCNH2GPR84HCAR2HCAR3CYP3A4
SCHEMBL27724995 0.98 KCNH2 (0.39) KCNH2GPR84HCAR2HCAR3CYP3A4
SCHEMBL21634151 0.98 KCNH2 (0.39) KCNH2GPR84HCAR2HCAR3CYP3A4
SCHEMBL11480358 0.98 KCNH2 (0.39) KCNH2GPR84HCAR2HCAR3CYP3A4
SCHEMBL7812120 0.98 KCNH2 (0.39) KCNH2GPR84HCAR2HCAR3CYP3A4
SCHEMBL5991669 0.93
SCHEMBL16673289 0.89 L3MBTL1 (0.37) L3MBTL1ALDH1A1
SCHEMBL9633268 0.88 EPHX2 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 68 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107286133-B Application of -5 (the 4H)-thioketones imines of 3- aryl -1,2,4- triazole as NA inhibitor 湖南大学 2019-05-10 CN claimed
CN-107286133-A (4H) the thioketones imines of 3 aryl, 1,2,4 triazole 5 as NA inhibitor application 湖南大学 2017-10-24 CN claimed
US-4814112-A Single-stage process for preparing mixed-substituted 1,2-diacyl-sn-clycero-3-phosphocholines CL PHARMA AKTIENGESELLSCHAFT (AT) 1989-03-21 US claimed
US-20250215572-A1 SURFACE TREATMENT AGENT FOR COPPER OR COPPER ALLOY SHIKOKU CHEMICALS CORPORATION (JP) 2025-07-03 US disclosed
EP-4506488-A1 SURFACE TREATMENT AGENT FOR COPPER OR COPPER ALLOY Shikoku Chemicals Corporation (JP) 2025-02-12 EP disclosed
CN-118922584-A Surface treating agent for copper or copper alloy 四国化成工业株式会社 2024-11-08 CN disclosed
WO-2023190263-A1 SURFACE TREATMENT AGENT FOR COPPER OR COPPER ALLOY 四国化成工業株式会社 2023-10-05 WO disclosed
EP-3834828-B1 COMPOSITION COMPRISING A THIAMINE DERIVATIVE FOR USE IN THE PREVENTION OR TREATMENT OF VASCULAR OR CARDIAC VALVE CALCIFICATION KYUNGPOOK NAT UNIV IND ACADEMIC COOP FOUND (KR) 2022-06-08 EP disclosed
US-11331317-B2 Composition for treating vascular or cardiac valvular calcification, containing thiamine derivative KYUNGPOOK NATIONAL UNIVERSITY INDUSTRY-ACADEMIC COOPERATION FOUNDATION (KR) 2022-05-17 US disclosed
US-20210290621-A1 COMPOSITION FOR PREVENTING OR TREATING VASCULAR OR CARDIAC VALVULAR CALCIFICATION, CONTAINING THIAMINE DERIVATIVE PRIMEMUPHARMA CO., LTD (KR) 2021-09-23 US disclosed
EP-3834828-A1 COMPOSITION FOR PREVENTING OR TREATING VASCULAR OR CARDIAC VALVULAR CALCIFICATION, CONTAINING THIAMINE DERIVATIVE Kyungpook National University Industry-Academic Cooperation Foundation (KR) 2021-06-16 EP disclosed
WO-1996018618-A1 3-ARYL-1,2,4-TRIAZOLE DERIVATIVES WITH HERBICIDAL PROPERTIES BAYER AKTIENGESELLSCHAFT (DE) 1996-06-20 WO disclosed
US-4888350-A ANTIFERTILITY AGENTS GRUPPO LEPETIT S.P.A. (IT) 1989-12-19 US disclosed
US-4888350-A ANTIFERTILITY AGENTS GRUPPO LEPETIT S.P.A. (IT) 1989-12-19 US disclosed
US-4888350-A ANTIFERTILITY AGENTS GRUPPO LEPETIT S.P.A. (IT) 1989-12-19 US disclosed
US-4459302-A CONTRACEPTIVES GRUPPO LEPETIT, S.P.A. (IT) 1984-07-10 US disclosed
US-4459302-A CONTRACEPTIVES GRUPPO LEPETIT, S.P.A. (IT) 1984-07-10 US disclosed
US-4459302-A CONTRACEPTIVES GRUPPO LEPETIT, S.P.A. (IT) 1984-07-10 US disclosed
US-4069035-A PLANT GROWTH REGULATORS, PICRATE DYES E. I. DU PONT DE NEMOURS AND COMPANY (US) 1978-01-17 US disclosed
US-4038285-A BUFFER SOLUTIONS, PICRATE DYES, PLANT GROWTH REGULATORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1977-07-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210290621-A1 COMPOSITION FOR PREVENTING OR TREATING VASCULAR OR CARDIAC VALVULAR CALCIFICATION, CONTAINING THIAMINE DERIVATIVE SLC19A2, FABP3, SLC5A6 KCNH2 421/4885GPR84 4014/4885HCAR2 1009/4885
US-11331317-B2 Composition for treating vascular or cardiac valvular calcification, containing thiamine derivative SLC19A2, VDR, SLC5A6 KCNH2 385/4885GPR84 3533/4885HCAR2 1100/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.