SCHEMBL10181022

SCHEMBL10181022

Cc1cccc(COc2ccc(Cl)cc2C(=O)NCCc2ccc(-c3ccc(OC(=O)O)cc3)cc2)c1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 5/20 0.57
DNMT3A Q9Y6K1 1/20 0.52
HDAC1 Q13547 3/20 0.46
HDAC6 Q9UBN7 3/20 0.46
NLRP3 Q96P20 3/20 0.46
KMT2A Q03164 1/20 0.46
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
THRB P10828 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10181905 0.91 DNMT3A (0.58) AKR1C3DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10181019 0.90 DNMT3A (0.56) AKR1C3DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10181047 0.90 AKR1C3 (0.51) AKR1C3DNMT3AHDAC1HDAC6NLRP3
SCHEMBL1154137 0.89 AKR1C3 (0.59) AKR1C3DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10181116 0.87 LRRK2 (0.50) AKR1C3DNMT3A
SCHEMBL10182099 0.86 DNMT3A (0.52) AKR1C3DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10181359 0.85 DNMT3A (0.53) AKR1C3DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10180516 0.85 LRRK2 (0.55) AKR1C3DNMT3AHDAC1HDAC6KMT2A
SCHEMBL10181121 0.85 DNMT3A (0.56) AKR1C3DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10182210 0.83 DNMT3A (0.54) AKR1C3DNMT3AHDAC1HDAC6NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2215065-B1 CCR10 ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-07-11 EP claimed