SCHEMBL10181047

SCHEMBL10181047

O=C(O)Oc1ccc(-c2ccc(CCNC(=O)c3cc(Cl)ccc3OCc3cccc(F)c3)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.51
DNMT3A Q9Y6K1 1/20 0.49
KMT2A Q03164 1/20 0.46
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
SNCA P37840 1/20 0.44
NLRP3 Q96P20 3/20 0.44
HIF1A Q16665 1/20 0.43
PTGER4 P35408 1/20 0.43
POLB P06746 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
MCHR1 Q99705 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10181359 0.91 DNMT3A (0.53) AKR1C3DNMT3AKMT2AHDAC1HDAC6
SCHEMBL10182099 0.90 DNMT3A (0.52) AKR1C3DNMT3AKMT2AHDAC1HDAC6
SCHEMBL10181022 0.90 AKR1C3 (0.57) AKR1C3DNMT3AKMT2AHDAC1HDAC6
SCHEMBL1154081 0.89 AKR1C3 (0.52) AKR1C3DNMT3AKMT2AHDAC1HDAC6
SCHEMBL10181116 0.89 LRRK2 (0.50) AKR1C3DNMT3A
SCHEMBL10181019 0.89 DNMT3A (0.56) AKR1C3DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10180506 0.86 AKR1C3 (0.51) AKR1C3DNMT3AKMT2AHDAC1HDAC6
SCHEMBL10181905 0.85 DNMT3A (0.58) AKR1C3DNMT3AHDAC1HDAC6NLRP3
SCHEMBL10180516 0.85 LRRK2 (0.55) AKR1C3DNMT3AKMT2AHDAC1HDAC6
SCHEMBL10181121 0.83 DNMT3A (0.56) AKR1C3DNMT3AKMT2AHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2215065-B1 CCR10 ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-07-11 EP claimed