SCHEMBL10183085

SCHEMBL10183085

CC(C)(C)c1cnn2cc(-c3cnc(N)nc3)ccc12

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 19/20 0.40
FEN1 P39748 3/20 0.40
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10182972 0.82 PIK3CG (0.37)
SCHEMBL10182956 0.81 JAK1 (0.38) MAPT
SCHEMBL10183055 0.79 KIF11 (0.44) LMNAMAPT
SCHEMBL10182958 0.75 KIF11 (0.50)
SCHEMBL10183063 0.75 KIT (0.32) MAPT
SCHEMBL10183057 0.75 BMP4 (0.37)
SCHEMBL10182971 0.75 JAK1 (0.40) MAPT
SCHEMBL10182940 0.73 JAK1 (0.38)
SCHEMBL10182985 0.73 MAP4K4 (0.49) ALOX5APLMNAMAPT
SCHEMBL10182966 0.73 ACVR2A (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120040951-A1 HETEROARYL COMPOUNDS USEFUL AS RAF KINASE INHIBITORS SUNESIS PHARMACEUTICALS, INC. 2012-02-16 US disclosed
US-20120040951-A1 HETEROARYL COMPOUNDS USEFUL AS RAF KINASE INHIBITORS SUNESIS PHARMACEUTICALS, INC. 2012-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120040951-A1 HETEROARYL COMPOUNDS USEFUL AS RAF KINASE INHIBITORS BRAF, RAF1, ARAF ALOX5AP 3549/4885FEN1 978/4885LMNA 3593/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.