SCHEMBL10187349

SCHEMBL10187349

Cc1ncc(-c2ccc3[nH]ccc3c2)cc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 4/20 0.52
LRRK2 Q5S007 4/20 0.50
BRD4 O60885 1/20 0.49
NPC1 O15118 1/20 0.49
AHR P35869 1/20 0.49
DYRK1A Q13627 2/20 0.47
DYRK2 Q92630 2/20 0.47
DYRK1B Q9Y463 2/20 0.47
CLK1 P49759 1/20 0.47
PIK3CD O00329 1/20 0.46
PIK3CA P42336 1/20 0.46
MTOR P42345 1/20 0.46
PIP4K2A P48426 1/20 0.45
PIP4K2B P78356 1/20 0.45
GUSB P08236 1/20 0.45
FYN P06241 1/20 0.45
CHRNA7 P36544 1/20 0.44
KCNH2 Q12809 1/20 0.44
ABL1 P00519 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19391087 0.80 DYRK1B (0.47) MAP3K11LRRK2NPC1AHRDYRK1A
SCHEMBL14365330 0.76 MAP3K11 (0.67) MAP3K11LRRK2NPC1DYRK1ADYRK2
SCHEMBL5850255 0.75 NPC1 (0.79) MAP3K11BRD4NPC1AHRGUSB
SCHEMBL16881490 0.74 BRD4 (0.47) LRRK2BRD4DYRK1ADYRK2DYRK1B
SCHEMBL20261213 0.74 ABL1 (0.49) CHRNA7KCNH2ABL1
SCHEMBL13354456 0.74 PIP4K2A (0.58) MAP3K11LRRK2BRD4NPC1DYRK1A
SCHEMBL857265 0.73 RIPK1 (0.57) LRRK2BRD4DYRK1ADYRK1BPIK3CD
SCHEMBL12680497 0.73 NPC1 (0.56) MAP3K11LRRK2NPC1AHRDYRK1A
SCHEMBL21250701 0.73 NPC1 (0.60) MAP3K11LRRK2NPC1DYRK1ADYRK2
SCHEMBL29475133 0.72 BRD4 (0.48) MAP3K11LRRK2BRD4NPC1AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012001107-A1 PIPERIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-05 WO disclosed