SCHEMBL10194199

SCHEMBL10194199

CS/C(N)=N\c1cccc2ncc(NC(=O)c3ccc(N)cn3)cc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 4/20 0.38
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPT P10636 1/20 0.36
ACKR3 P25106 1/20 0.36
KDR P35968 5/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
POLB P06746 1/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
BLK P51451 1/20 0.35
MITF O75030 1/20 0.34
XBP1 P17861 1/20 0.34
PAX8 Q06710 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10194914 0.87 ALDH1A1 (0.43) ALDH1A1KDM4ENPC1RAB9AHPGD
SCHEMBL10192946 0.87 BACE1 (0.42)
SCHEMBL10194907 0.86 SMN1; SMN2 (0.38) ALDH1A1NPC1RAB9AMAPTACKR3
SCHEMBL10193944 0.77 KDM4E (0.43) ALDH1A1KDM4ENPC1RAB9AHPGD
SCHEMBL10193263 0.74 ALDH1A1 (0.48) ALDH1A1KDM4ENPC1RAB9AHPGD
SCHEMBL10193577 0.74 RAB9A (0.38) ALDH1A1KDM4ENPC1RAB9AMAPT
SCHEMBL10193848 0.74 BACE1 (0.43) ALDH1A1KDM4ENPC1RAB9AHPGD
SCHEMBL10193028 0.73 BACE1 (0.44) ALDH1A1KDM4ENPC1RAB9AHPGD
SCHEMBL10192941 0.73 BACE1 (0.44)
SCHEMBL10193707 0.73 PDE4D (0.42) ALDH1A1KDM4ENPC1RAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415756-A1 ISOTHIOUREA DERIVATIVES OR ISOUREA DERIVATIVES HAVING BACE1 INHIBITORY ACTIVITY Shionogi&Co., Ltd. (JP) 2012-02-08 EP disclosed