SCHEMBL10194913

SCHEMBL10194913

N=C(c1cn(-c2cccc(CCCN3CCOCC3)c2)nn1)c1ccccc1N

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESRRA P11474 11/20 0.49
FAAH O00519 1/20 0.47
MGLL Q99685 1/20 0.47
SIGMAR1 Q99720 3/20 0.43
POLB P06746 1/20 0.43
MAPK14 Q16539 1/20 0.41
HTR7 P34969 2/20 0.41
DDX3X O00571 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10194915 0.92 ESRRA (0.52) ESRRAFAAHMGLLSIGMAR1HTR7
SCHEMBL10196715 0.86 ESRRA (0.53) ESRRAFAAHMGLLSIGMAR1
SCHEMBL10194711 0.78 ESRRA (0.60) ESRRAFAAHMGLL
SCHEMBL10195783 0.78 ESRRA (0.55) ESRRAFAAHMGLL
SCHEMBL10195750 0.76 ESRRA (0.62) ESRRAFAAHMGLL
SCHEMBL10196894 0.75 ESRRA (0.56) ESRRAFAAHMGLLPOLB
SCHEMBL10194732 0.73 ESRRA (0.44) ESRRA
SCHEMBL10195780 0.73 ESRRA (0.44) ESRRA
SCHEMBL17850412 0.71 ESRRA (0.48) ESRRA
SCHEMBL10194692 0.70 SIGMAR1 (0.44) FAAHMGLLSIGMAR1POLBHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012084704-A1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO S.A. (CH) 2012-06-28 WO disclosed