SCHEMBL10195044

SCHEMBL10195044

CO/C(N)=N/C(c1cccc(F)c1)c1cccc(NC(=O)c2ccc(N)cn2)c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.45
KDM4E B2RXH2 1/20 0.43
HDAC3 O15379 6/20 0.41
HDAC1 Q13547 6/20 0.41
HDAC2 Q92769 6/20 0.41
NCOR2 Q9Y618 6/20 0.41
BACE1 P56817 3/20 0.40
ALDH1A1 P00352 2/20 0.39
POLB P06746 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
ACKR3 P25106 1/20 0.39
AURKA O14965 2/20 0.39
RPS6KB1 P23443 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10194093 0.91 BACE1 (0.42) SMN1; SMN2KDM4EHDAC3HDAC1HDAC2
SCHEMBL10193694 0.88 SMN1; SMN2 (0.48) SMN1; SMN2KDM4EBACE1ALDH1A1MEN1
SCHEMBL10193565 0.88 ALDH1A1 (0.39) SMN1; SMN2HDAC3HDAC1HDAC2NCOR2
SCHEMBL10194892 0.88 AURKA (0.43) SMN1; SMN2KDM4EALDH1A1MEN1KMT2A
SCHEMBL10193931 0.87 BACE1 (0.46) BACE1
SCHEMBL10193709 0.86 SMN1; SMN2 (0.42) SMN1; SMN2BACE1ALDH1A1POLBMEN1
SCHEMBL10193160 0.81 BACE1 (0.48) SMN1; SMN2BACE1ALDH1A1POLBMEN1
SCHEMBL10193843 0.81 BACE1 (0.45) BACE1
SCHEMBL10193937 0.81 BACE1 (0.45) BACE1
SCHEMBL10193017 0.78 BACE1 (0.47) BACE1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415756-A1 ISOTHIOUREA DERIVATIVES OR ISOUREA DERIVATIVES HAVING BACE1 INHIBITORY ACTIVITY Shionogi&Co., Ltd. (JP) 2012-02-08 EP disclosed