SCHEMBL10195751

SCHEMBL10195751

COC(=O)c1ccc(-n2cc(C(=N)c3cc(C)ccc3NC(=O)OC(C)(C)C)nn2)cc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESRRA P11474 1/20 0.40
PSMD10 O75832 1/20 0.40
CA1 P00915 4/20 0.39
CA2 P00918 4/20 0.39
CA9 Q16790 4/20 0.39
CA12 O43570 3/20 0.39
NOTUM Q6P988 3/20 0.39
CA4 P22748 1/20 0.38
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KMT2A Q03164 1/20 0.37
P2RY14 Q15391 1/20 0.37
GPR119 Q8TDV5 3/20 0.36
DDT P30046 2/20 0.36
AURKA O14965 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10195752 0.76 GPR119 (0.40) CA1CA2CA9CA12CA4
SCHEMBL31227601 0.69 PSMD10 (0.52) ESRRAPSMD10CA1CA2CA9
SCHEMBL25241550 0.69 CA1 (0.48) PSMD10CA1CA2CA9CA12
SCHEMBL10194877 0.68 HPGD (0.44) CA1CA9CA12POLBKMT2A
SCHEMBL12393084 0.68 GLA (0.51) CA1CA2CA9CA12CA4
SCHEMBL12393083 0.68 MIF (0.53) CA1CA2CA9CA12POLB
SCHEMBL21997183 0.68 LCK (0.37) CA1CA2CA9CA12POLB
SCHEMBL4502703 0.67 KDM4E (0.48) L3MBTL1KMT2A
SCHEMBL11959276 0.67 LCK (0.49) CA1CA2CA9CA12NOTUM
SCHEMBL27852761 0.67 MEN1 (0.56) CA1CA12CA4L3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012084704-A1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO S.A. (CH) 2012-06-28 WO disclosed