SCHEMBL10200000

SCHEMBL10200000

CC(C)(Oc1ccc(O)c(O)c1)C(=O)Nc1ncc(Cl)s1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
FFAR2 O15552 3/20 0.44
POLB P06746 1/20 0.44
GCK P35557 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP2D6 P10635 1/20 0.42
ADORA2A P29274 3/20 0.42
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2657244 0.82 GCK (0.55) ALDH1A1FFAR2POLBGCKCYP1A2
SCHEMBL2658792 0.82 NPC1 (0.52) ALDH1A1FFAR2POLBGCKCYP1A2
SCHEMBL2661038 0.81 ADORA2A (0.56) POLBADORA2A
SCHEMBL2656942 0.81 ALDH1A1 (0.50) ALDH1A1FFAR2POLBGCKCYP1A2
SCHEMBL2656485 0.81 GCK (0.47) ALDH1A1FFAR2POLBGCKADORA2A
SCHEMBL2662251 0.81 POLB (0.42) ALDH1A1FFAR2POLBGCKCYP1A2
SCHEMBL2656521 0.81 POLB (0.60) ALDH1A1FFAR2POLBGCKCYP1A2
SCHEMBL2657292 0.80 CYP1A2 (0.43) ALDH1A1FFAR2POLBGCKCYP1A2
SCHEMBL2655818 0.80 FFAR2 (0.45) ALDH1A1FFAR2POLBGCKCYP1A2
SCHEMBL2657121 0.79 CYP1A2 (0.45) ALDH1A1FFAR2POLBGCKCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125735-B1 2,2,2-TRI-SUBSTITUTED ACETAMIDE DERIVATIVES AS GLUCOKINASE ACTIVATORS, THEIR PROCESS AND PHARMACEUTICAL APPLICATION ADVINUS THERAPEUTICS PRIVATE LTD (IN) 2012-06-27 EP disclosed