SCHEMBL10200872

SCHEMBL10200872

Cc1cncc2cncnc12

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.37
CCR1 P32246 1/20 0.33
CCR5 P51681 1/20 0.33
CCR8 P51685 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31610186 1.00 EGFR (0.37) EGFRCCR1CCR5CCR8CYP1A2
SCHEMBL2843194 0.76 EGFR (0.47) EGFRCYP1A2CYP3A4CYP2D6
SCHEMBL8404389 0.76 CCR1 (0.39) EGFRCCR1CCR5CCR8CYP1A2
SCHEMBL24495971 0.74 CCR1 (0.32) CCR1CCR5CCR8
SCHEMBL18266950 0.74 CCR1 (0.58) CCR1CCR5CCR8CYP1A2
Benzene SCHEMBL27961712 0.74 EGFR (0.45) EGFRCYP1A2CYP3A4CYP2D6
SCHEMBL22915040 0.73 EGFR (0.34) EGFR
SCHEMBL24464882 0.73 NQO2 (0.41) EGFR
SCHEMBL24857275 0.71 EGFR (0.37) EGFR
SCHEMBL3239463 0.71 EGFR (0.37) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023110138-A1 INHIBITORS OF TRANSGLUTAMINASES ZEDIRA GMBH (DE) 2023-06-22 WO disclosed
WO-2016118823-A1 PTERIDINE DIONE MONOCARBOXYLATE TRANSPORTER INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 2016-07-28 WO disclosed
WO-2016118822-A1 CHROMENONE INHIBITORS OF MONOCARBOXYLATE TRANSPORTERS THE SCRIPPS RESEARCH INSTITUTE (US) 2016-07-28 WO disclosed
US-20120030841-A1 Isoxazoline compounds for combating invertebrate pests BASF SE (DE) 2012-02-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120030841-A1 Isoxazoline compounds for combating invertebrate pests PRDX5, PRDX1, PRDX2 EGFR 4875/4885CCR1 4384/4885CCR5 3366/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.