SCHEMBL24464882

SCHEMBL24464882

Cc1cc(Br)cc2cncnc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 2/20 0.41
EGFR P00533 9/20 0.36
PRNP P04156 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
NOD2 Q9HC29 1/20 0.33
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
PARP4 Q9UKK3 1/20 0.31
EGLN1 Q9GZT9 1/20 0.31
GSK3A P49840 1/20 0.30
CDK9 P50750 1/20 0.30
CDK5 Q00535 1/20 0.30
TAOK1 Q7L7X3 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8404389 0.80 CCR1 (0.39) EGFRLMNAHPGDHTTALDH1A1
SCHEMBL29550394 0.77 TRPV1 (0.33) EGFRGSK3ACDK9CDK5TAOK1
SCHEMBL30902155 0.77 EGFR (0.32) EGFREGLN1GSK3ACDK9CDK5
SCHEMBL19878479 0.77 NQO2 (0.45) NQO2EGFRPRNPNPSR1ALDH1A1
SCHEMBL31716595 0.74 SMN1; SMN2 (0.38) NQO2PRNPNPSR1LMNAHPGD
SCHEMBL3928379 0.73 CCR1 (0.36) NQO2EGFRPRNPNPSR1LMNA
SCHEMBL38659591 0.73 SRC (0.34) EGFR
SCHEMBL31610506 0.73 HPGDS (0.39) EGFRLMNAHTTALDH1A1L3MBTL1
SCHEMBL29439776 0.73 EPRS1 (0.35) ALDH1A1
SCHEMBL10200872 0.73 EGFR (0.37) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4006035-A1 QUINAZOLINE DERIVATIVES AS TYROSINE KINASE INHIBITORS FOR THE TREATMENT OF CANCER Neupharma, Inc. (US) 2022-06-01 EP disclosed