SCHEMBL10201035

SCHEMBL10201035

CC(C)(C(=O)O)C(c1cccc(F)c1)c1ccc(N2CCCCC2)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 1/20 0.39
SLC6A2 P23975 3/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
SLC6A3 Q01959 1/20 0.37
SMN1; SMN2 Q16637 4/20 0.37
DPP4 P27487 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
TSHR P16473 2/20 0.34
MAPK1 P28482 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
TP53 P04637 3/20 0.33
MAPT P10636 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10201034 0.90 KCNQ2 (0.40) KCNQ2SLC6A2CHRNB2CHRNB4CHRNA3
SCHEMBL753423 0.90 AR (0.40) SMN1; SMN2DPP4DPP7MAPK1TP53
SCHEMBL752315 0.80 MAPT (0.40) SMN1; SMN2MAPTNPC1RAB9AADORA2A
SCHEMBL10331383 0.78 HDAC4 (0.40) SMN1; SMN2DPP4DPP7OPRM1
SCHEMBL14207656 0.78 HDAC4 (0.37) DPP4DPP7OPRM1
SCHEMBL10331384 0.78 HDAC4 (0.40) SMN1; SMN2DPP4DPP7OPRM1
SCHEMBL754423 0.78 HDAC4 (0.40) SMN1; SMN2DPP4DPP7OPRM1
SCHEMBL14207516 0.72 MAPT (0.34) SMN1; SMN2MAPTNPC1RAB9AADORA2A
SCHEMBL753470 0.72 NR3C1 (0.50)
SCHEMBL751383 0.72 NR3C1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078015-B1 MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1 AND/OR NF-KAPPAB ACTIVITY AND USE THEREOF BRISTOL MYERS SQUIBB CO (US) 2012-03-21 EP disclosed