SCHEMBL1020908

SCHEMBL1020908

NC(=O)c1ccc(C(=O)NC2=NCCO2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.43
RAB9A P51151 5/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
CASP3 P42574 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
KMT2A Q03164 3/20 0.41
MAPT P10636 2/20 0.41
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
CCNA1 P78396 1/20 0.41
TSHR P16473 1/20 0.39
KDM4E B2RXH2 4/20 0.38
MEN1 O00255 2/20 0.38
BCAT2 O15382 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
PLAU P00749 2/20 0.36
F2 P00734 1/20 0.36
PLG P00747 1/20 0.36
KLKB1 P03952 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31692769 0.84 NPC1 (0.48) NPC1RAB9ASMN1; SMN2KMT2AKDM4E
SCHEMBL27768543 0.77
SCHEMBL6591819 0.72 LSS (0.46) NPC1RAB9ASMN1; SMN2CASP3SENP7
SCHEMBL28294378 0.69
SCHEMBL13210699 0.68 KMT2A (0.73) NPC1RAB9ASMN1; SMN2CASP3SENP7
Sulfuric Acid SCHEMBL11149992 0.66 ADRA2A (0.35) MAPTTSHRKDM4ECYP2C9POLB
SCHEMBL28872262 0.65 CYP3A4 (0.42) MAPTTSHRKDM4ECYP2C9POLB
SCHEMBL1664024 0.65 MEN1 (0.59) NPC1RAB9AKMT2AMAPTTSHR
SCHEMBL28829404 0.65 KDM4E (0.81) NPC1RAB9ASMN1; SMN2KMT2AMAPT
Terephthalamide SCHEMBL23774 0.64 PARP1 (0.71) SMN1; SMN2KMT2AMAPTTSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271642-A2 PYRIDYL INHIBITORS OF HEDGEHOG SIGNALLING Genentech, Inc. (US) 2011-01-12 EP disclosed