SCHEMBL1020975

SCHEMBL1020975

COc1cccc(N(F)F)c1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.42
CA2 P00918 4/20 0.42
CA7 P43166 3/20 0.42
CA9 Q16790 3/20 0.42
CA12 O43570 2/20 0.42
CA14 Q9ULX7 2/20 0.42
CA4 P22748 1/20 0.42
ALDH1A1 P00352 3/20 0.39
TP53 P04637 2/20 0.39
MAPK1 P28482 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
HSD17B10 Q99714 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.36
NFE2L2 Q16236 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27665453 0.81 TUBB1 (0.35) CA1CA2CA7CA9CA12
SCHEMBL4302129 0.80 CA1 (0.55) CA1CA2CA7CA9CA12
SCHEMBL630768 0.79 CA1 (0.58) CA1CA2CA7CA9CA12
SCHEMBL2094827 0.74 CA1 (0.46) CA1CA2CA7CA9CA12
SCHEMBL10578058 0.73 TUBB1 (0.35) CA1CA2CA7CA9CA12
SCHEMBL27759581 0.73 TUBB1 (0.33) CA1CA2CA7CA9CA12
SCHEMBL196734 0.73 CA1 (0.50) CA1CA2CA7CA9CA12
SCHEMBL29387155 0.73 CA1 (0.50) CA1CA2CA7CA9CA12
SCHEMBL11016571 0.72 RAB9A (0.34) CA1CA2CA7CA9CA12
SCHEMBL5633423 0.72 TUBB1 (0.33) CA1CA2CA7CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 94 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109678788-A A kind of 1,2- diaryl indoles, derivative and its synthetic method 湘潭大学 2019-04-26 CN claimed
CN-106946781-B A kind of pyrazoles diphenyl urea analog derivative and its preparation method and application 合肥工业大学 2019-04-19 CN claimed
CN-107032965-A A kind of preparation method of 3 trifluoro-methoxy-phenol 金凯(辽宁)化工有限公司 2017-08-11 CN claimed
CN-102797043-B Medicinal molecular fragment library and construction process thereof Tianli (Tianjin) Technology Co., Ltd. (CN) 2015-11-25 CN claimed
CN-104262181-A Preparing method of fluorine-group-containing ethyl 3-(phenyl-1-imine) propionate analogues SHANGHAI INST TECHNOLOGY 2015-01-07 CN claimed
CN-102797043-A Medicinal molecular fragment library and construction method thereof CBB NETWORK CO LTD 2012-11-28 CN claimed
CN-109678788-A A kind of 1,2- diaryl indoles, derivative and its synthetic method 湘潭大学 2019-04-26 CN disclosed
CN-106946781-B A kind of pyrazoles diphenyl urea analog derivative and its preparation method and application 合肥工业大学 2019-04-19 CN disclosed
CN-108047142-A Heteroaryl compound and its purposes 阿维拉制药公司 2018-05-18 CN disclosed
CN-104892485-B 2 perfluoroalkyl indole derivativeses and its synthetic method 上海麦克林生化科技有限公司 2018-03-23 CN disclosed
CN-107108536-A Biguanide compound and application thereof 伊谬诺米特医疗有限公司 2017-08-29 CN disclosed
CN-107098846-A N- acyl sulfonamides class FBPase inhibitor, its preparation method, pharmaceutical composition and purposes 中国医学科学院药物研究所 2017-08-29 CN disclosed
CN-107032965-A A kind of preparation method of 3 trifluoro-methoxy-phenol 金凯(辽宁)化工有限公司 2017-08-11 CN disclosed
CN-1043531-C Pyrimidine derivatives and a process for production thereof NOVATIS AG (CH) 1999-06-02 CN disclosed
EP-0862560-A1 SUBSTITUTED 2-ANILINOPYRIMIDINES USEFUL AS PROTEIN KINASE INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 1998-09-09 EP disclosed
CN-1190962-A Process for the preparation of substituted 5-hydroxy-oxazolidin-4-one ZENECA LTD (GB) 1998-08-19 CN disclosed
WO-1997019065-A1 SUBSTITUTED 2-ANILINOPYRIMIDINES USEFUL AS PROTEIN KINASE INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 1997-05-29 WO disclosed
CN-1092425-A Indole derivatives, its manufacture method and medicinal use thereof TORAY INDUSTRIES (JP) 1994-09-21 CN disclosed
CN-1077713-A Pyrimidine derivatives and preparation method thereof CIBA GEIGY AG (CH) 1993-10-27 CN disclosed
CN-1074678-A 1, the 5-benzodiazepine derivatives GLAXO SPA (IT) 1993-07-28 CN disclosed