SCHEMBL1021653

SCHEMBL1021653

CCCCC1=C(c2cccc(C)c2)C(=O)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
SIRT2 Q8IXJ6 5/20 0.37
SIRT1 Q96EB6 3/20 0.36
PGR P06401 1/20 0.36
TP53 P04637 1/20 0.36
PARP10 Q53GL7 1/20 0.35
PARP11 Q9NR21 1/20 0.35
TLR8 Q9NR97 1/20 0.35
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
FYN P06241 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1022356 0.84 BRD4 (0.40)
SCHEMBL1020035 0.84 ESR1 (0.40)
SCHEMBL1021433 0.84 NPC1 (0.36) CHRNB4CHRNA3MAPTCTSSCTSK
SCHEMBL1021866 0.82 CHRNB4 (0.38) PGRCHRNB4CHRNA3
SCHEMBL1022920 0.82 BRD4 (0.42) TLR8
SCHEMBL1025827 0.81 PTPN11 (0.44)
SCHEMBL1020478 0.81 MAPT (0.45) KDM4ETP53MAPT
SCHEMBL1021059 0.81 TLR8 (0.40) PARP10PARP11TLR8CTSSCTSK
SCHEMBL1022880 0.81 BRD4 (0.39) KDM4ETP53MAPTHTTCTSK
SCHEMBL1021652 0.81 PTGS1 (0.48) TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1841729-B1 2-CYCLOPENTEN-1-ONE OXIME DERIVATIVES INHIBITING PRODUCTION OF TNF-ALPHA AMOREPACIFIC CORP (KR) 2011-01-12 EP claimed