SCHEMBL1021865

SCHEMBL1021865

CC(C)(C)COC(=O)N(OC(=O)C(F)(F)F)c1ccc(C(=O)N2CCN(Cc3cccc(C(=O)NC(C)(C)C)c3)CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 5/20 0.41
LMNA P02545 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
GAA P10253 1/20 0.41
MEN1 O00255 5/20 0.40
KMT2A Q03164 5/20 0.40
SIGMAR1 Q99720 1/20 0.40
MAPT P10636 1/20 0.40
RECQL P46063 1/20 0.40
MAPK1 P28482 2/20 0.39
TSHR P16473 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ACKR3 P25106 2/20 0.38
LSS P48449 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM3 P20309 1/20 0.38
HTT P42858 1/20 0.38
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1075172 0.90 ACKR3 (0.40) KDM4EALDH1A1LMNASMN1; SMN2GAA
Trifluoroacetic Acid SCHEMBL1021864 0.81 PRKAB2 (0.47) KDM4EALDH1A1LMNASMN1; SMN2GAA
SCHEMBL1017900 0.77 MEN1 (0.53) KDM4EALDH1A1LMNASMN1; SMN2GAA
SCHEMBL3688234 0.74 CHRM2 (0.46) KDM4EALDH1A1LMNASMN1; SMN2GAA
SCHEMBL28052665 0.74 MEN1 (0.53) KDM4EALDH1A1LMNASMN1; SMN2GAA
Trifluoroacetic Acid SCHEMBL1018638 0.74 PRKAB2 (0.48) KDM4EALDH1A1LMNASMN1; SMN2GAA
SCHEMBL1019016 0.73 SMN1; SMN2 (0.54) KDM4EALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL1018777 0.73 MEN1 (0.57) KDM4EALDH1A1LMNASMN1; SMN2GAA
SCHEMBL1023329 0.73 HPGD (0.45) KDM4EALDH1A1LMNASMN1; SMN2GAA
Trifluoroacetic Acid SCHEMBL1075170 0.73 BCHE (0.49) KDM4EALDH1A1LMNASMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190827-B1 N-BENZYL-N'-ARYLCARBONYLPIPERAZINE DERIVATIVES AS LXR MODULATORS ORGANON NV (NL) 2011-01-12 EP disclosed
EP-2190827-A1 N-BENZYL, N' -ARYLCARBONYLPIPERAZINE DERIVATIVES AS LXR MODULATORS N.V. Organon (NL) 2010-06-02 EP disclosed
WO-2009024550-A1 N-BENZYL, N' -ARYLCARBONYLPIPERAZINE DERIVATIVES AS LXR MODULATORS N.V. ORGANON (NL) 2009-02-26 WO disclosed