SCHEMBL10241635

SCHEMBL10241635

CCC1/C=C(\C)C[C@H](C)C[C@H](OC)[C@H]2O[C@@](O)(C(=O)C(=O)N3CCCC[C@H]3C(=O)O[C@H](/C(C)=C/[C@@H]3CC[C@H](Cl)[C@H](OC)C3)[C@H](C)[C@@H](C)CC1=O)[C@H](C)C[C@@H]2OC

nearest known ligand 0.92

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.92
ADORA3 P0DMS8 1/20 0.92
FKBP1A P62942 18/20 0.83
MEN1 O00255 1/20 0.83
LMNA P02545 1/20 0.83
MAPT P10636 1/20 0.83
KMT2A Q03164 1/20 0.83
THRB P10828 1/20 0.83
FKBP4 Q02790 1/20 0.83
PPP3CA Q08209 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pimecrolimus SCHEMBL15277958 0.96 ABCB11 (1.00) ABCB11ADORA3FKBP1AMEN1LMNA
Pimecrolimus SCHEMBL26411 0.96 ABCB11 (1.00) ABCB11ADORA3FKBP1AMEN1LMNA
Pimecrolimus SCHEMBL4651515 0.96 ABCB11 (1.00) ABCB11ADORA3FKBP1AMEN1LMNA
Pimecrolimus SCHEMBL9947518 0.96 ABCB11 (1.00) ABCB11ADORA3FKBP1AMEN1LMNA
Pimecrolimus SCHEMBL117937 0.96 ABCB11 (1.00) ABCB11ADORA3FKBP1AMEN1LMNA
Pimecrolimus SCHEMBL436549 0.96 ABCB11 (1.00) ABCB11ADORA3FKBP1AMEN1LMNA
Pimecrolimus SCHEMBL438880 0.96 ABCB11 (1.00) ABCB11ADORA3FKBP1AMEN1LMNA
Pimecrolimus SCHEMBL4456276 0.96 ABCB11 (1.00) ABCB11ADORA3FKBP1AMEN1LMNA
Pimecrolimus SCHEMBL8194907 0.96 ABCB11 (1.00) ABCB11ADORA3FKBP1AMEN1LMNA
Pimecrolimus SCHEMBL10241642 0.96 ABCB11 (1.00) ABCB11ADORA3FKBP1AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8173840-B2 Compounds with high therapeutic index SIGNATURE R&D HOLDINGS, LLC (US) 2012-05-08 US disclosed