SCHEMBL10241861

SCHEMBL10241861

NC1(c2ccc(Br)cc2)CC(F)(F)C1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.35
KDM1A O60341 3/20 0.33
RCOR1 Q9UKL0 3/20 0.33
ALDH1A1 P00352 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPK1 P28482 1/20 0.33
MEN1 O00255 1/20 0.33
RAD52 P43351 1/20 0.33
KMT2A Q03164 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
BACE1 P56817 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22380426 0.77 MAOB (0.54) MAOAMAOB
SCHEMBL991567 0.77 CYP2A6 (0.42) CYP2A6KDM1ARCOR1ALDH1A1ALOX15
SCHEMBL24698364 0.76 MAOB (0.42) CYP2A6KDM1ARCOR1ALDH1A1ALOX15
SCHEMBL15401384 0.75 TAAR1 (0.39) CYP2A6KDM1ARCOR1TAAR1
SCHEMBL15401382 0.75 TAAR1 (0.39) CYP2A6KDM1ARCOR1TAAR1
Hydrochloric Acid SCHEMBL5060581 0.75 KDM1A (0.40) CYP2A6KDM1ARCOR1ALDH1A1ALOX15
SCHEMBL237630 0.74 TAAR1 (0.34) CYP2A6KDM1ARCOR1ALDH1A1ALOX15
SCHEMBL2038191 0.74 TAAR1 (0.34) CYP2A6KDM1ARCOR1ALDH1A1ALOX15
SCHEMBL24510105 0.74 SLC6A3 (0.43) MEN1RAD52KMT2ATAAR1MAOA
SCHEMBL9966307 0.73 AKT1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027322-A1 OXADIAZOLE INHIBITORS OF LEUKOTRIENE PRODUCTION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-03-01 WO disclosed