SCHEMBL10242715

SCHEMBL10242715

COc1cc2c(Oc3cc4sc(N)nc4cc3F)ccnc2cc1O

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 2/20 0.43
PDGFRA P16234 2/20 0.40
PDGFRB P09619 1/20 0.40
AXL P30530 4/20 0.40
MET P08581 4/20 0.40
KDR P35968 1/20 0.39
SRC P12931 1/20 0.39
TGFBR1 P36897 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL371554 0.92 FGFR2 (0.48) FGFR2PDGFRAPDGFRBAXLKDR
SCHEMBL20525612 0.80 ILK (0.38) FGFR2
SCHEMBL4575949 0.79 AXL (0.57) FGFR2PDGFRAPDGFRBAXLMET
SCHEMBL4591188 0.79 FGFR2 (0.51) FGFR2PDGFRAPDGFRBSRCTGFBR1
Bromide SCHEMBL15918462 0.78 AXL (0.56) FGFR2PDGFRAPDGFRBAXLMET
SCHEMBL5707550 0.78 CYP3A4 (0.53) AXL
SCHEMBL24444554 0.77 MET (0.43) PDGFRAPDGFRBAXLMETKDR
Hydrochloric Acid SCHEMBL5707606 0.77 CYP3A4 (0.51) AXL
SCHEMBL24444616 0.76 MET (0.58) PDGFRAPDGFRBAXLMETKDR
SCHEMBL13787639 0.76 SRC (0.61) FGFR2PDGFRAPDGFRBAXLMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2409704-A2 c-Met modulators and methods of use Exelixis Inc. (US) 2012-01-25 EP disclosed
EP-2392565-A1 c-Met modulators and methods of use Exelixis Inc. (US) 2011-12-07 EP disclosed
EP-2392564-A1 c-Met modulators and methods of use Exelixis Inc. (US) 2011-12-07 EP disclosed