SCHEMBL10253118

SCHEMBL10253118

CCCCc1ccc(N=CC=O)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.58
CYP2D6 P10635 2/20 0.58
CYP2C9 P11712 2/20 0.58
ALDH1A1 P00352 3/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 2/20 0.44
THRA P10827 2/20 0.44
THRB P10828 2/20 0.44
CA2 P00918 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CA1 P00915 1/20 0.42
RARB P10826 1/20 0.41
PLK1 P53350 1/20 0.41
CYP4Z1 Q86W10 2/20 0.40
CYP4F11 Q9HBI6 1/20 0.40
CYP4F12 Q9HCS2 1/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13524725 0.82 CYP3A4 (0.58) CYP3A4CYP2D6CYP2C9ALDH1A1HPGD
SCHEMBL14430275 0.81 CYP3A4 (0.68) CYP3A4CYP2D6CYP2C9ALDH1A1HSD17B10
SCHEMBL13805424 0.81 CYP2C9 (0.53) CYP3A4CYP2D6CYP2C9ALDH1A1HPGD
SCHEMBL5680616 0.80 CYP3A4 (0.66) CYP3A4CYP2D6CYP2C9ALDH1A1HSD17B10
SCHEMBL5678389 0.80 CYP3A4 (0.66) CYP3A4CYP2D6CYP2C9ALDH1A1HSD17B10
SCHEMBL5921414 0.80 CYP3A4 (0.66) CYP3A4CYP2D6CYP2C9ALDH1A1HSD17B10
SCHEMBL5920334 0.80 CYP3A4 (0.66) CYP3A4CYP2D6CYP2C9ALDH1A1HSD17B10
SCHEMBL5518344 0.78 CYP3A4 (0.53) CYP3A4CYP2D6CYP2C9ALDH1A1HPGD
SCHEMBL13590026 0.77 CYP3A4 (0.50) CYP3A4CYP2D6CYP2C9ALDH1A1HPGD
SCHEMBL11524101 0.76 CYP3A4 (0.60) CYP3A4CYP2D6CYP2C9ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8173638-B2 Compounds which modulate the CB2 receptor BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-05-08 US disclosed